SCHEMBL2171623

SCHEMBL2171623

NC(=O)C(Cc1ccc(Oc2ccc(F)cc2)cc1)NC(=O)Cc1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 4/20 0.57
LTA4H P09960 1/20 0.56
EPHX2 P34913 1/20 0.56
GPR34 Q9UPC5 2/20 0.56
SCN9A Q15858 2/20 0.54
CNR2 P34972 1/20 0.53
ITGB3 P05106 1/20 0.53
ITGA2B P08514 1/20 0.53
FCER2 P06734 2/20 0.52
MMP3 P08254 1/20 0.52
MMP9 P14780 1/20 0.52
ALDH1A1 P00352 3/20 0.51
CYP3A4 P08684 2/20 0.51
CYP2C19 P33261 2/20 0.51
KDM4E B2RXH2 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
PTPN2 P17706 2/20 0.50
PTPRA P18433 1/20 0.50
PTPN6 P29350 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2352923 0.87 SCN9A (0.64) PTPN1GPR34SCN9AFCER2MMP3
SCHEMBL5645893 0.85 PTPN1 (0.64) PTPN1CNR2ITGB3ITGA2BFCER2
SCHEMBL3956755 0.85 PTPN1 (0.64) PTPN1CNR2ITGB3ITGA2BFCER2
SCHEMBL2356381 0.85 SCN9A (0.50) PTPN1LTA4HEPHX2GPR34SCN9A
SCHEMBL2357204 0.84 SCN9A (0.52) PTPN1LTA4HEPHX2GPR34SCN9A
SCHEMBL2172994 0.81 POLB (0.52) GPR34SCN9AFCER2MMP3MMP9
SCHEMBL2170811 0.80 MAPT (0.54) SCN9AALDH1A1KDM4E
SCHEMBL2171096 0.79 SCN9A (0.51) LTA4HGPR34SCN9AALDH1A1KDM4E
SCHEMBL2353034 0.79 SCN9A (0.48) GPR34SCN9AITGB3ITGA2BFCER2
SCHEMBL2172340 0.79 SCN9A (0.51) GPR34SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346821-A1 SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS Exelixis, Inc. (US) 2011-07-27 EP disclosed