SCHEMBL2172994

SCHEMBL2172994

NC(=O)C(Cc1ccc(Oc2ccc(F)cc2)cc1)NC(=O)CN1Cc2ccccc2C1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.52
SCN9A Q15858 7/20 0.51
GPR34 Q9UPC5 2/20 0.44
ALDH1A1 P00352 1/20 0.43
FCER2 P06734 1/20 0.42
MMP3 P08254 1/20 0.42
MMP9 P14780 1/20 0.42
FPR1 P21462 2/20 0.41
FPR2 P25090 2/20 0.41
PRMT5 O14744 1/20 0.41
WDR77 Q9BQA1 1/20 0.41
TACR2 P21452 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2171096 0.86 SCN9A (0.51) POLBSCN9AGPR34ALDH1A1
SCHEMBL2170811 0.84 MAPT (0.54) POLBSCN9AALDH1A1
SCHEMBL2171621 0.83 QRFPR (0.50) SCN9AGPR34ALDH1A1
SCHEMBL2169808 0.83 SCN9A (0.48) SCN9AGPR34ALDH1A1TACR2
SCHEMBL2171851 0.83 KMT2A (0.53) SCN9AALDH1A1TACR2
SCHEMBL2170332 0.82 ALDH1A1 (0.53) SCN9AALDH1A1
SCHEMBL2170108 0.82 LMNA (0.52) POLBSCN9AALDH1A1
SCHEMBL2170398 0.82 ALDH1A1 (0.51) SCN9AALDH1A1
SCHEMBL2170433 0.82 SCN9A (0.47) SCN9AGPR34ALDH1A1FCER2MMP3
SCHEMBL2169958 0.82 SCN9A (0.47) SCN9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346821-A1 SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS Exelixis, Inc. (US) 2011-07-27 EP disclosed