SCHEMBL21723893

SCHEMBL21723893

COc1ccc(Cl)cc1/C=N/[S+]([O-])C(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.41
MAPT P10636 3/20 0.41
KDM4E B2RXH2 2/20 0.41
HPGD P15428 3/20 0.40
TSHR P16473 2/20 0.40
MEN1 O00255 3/20 0.37
ALDH1A1 P00352 2/20 0.37
MGAM O43451 1/20 0.36
GAA P10253 1/20 0.36
SI P14410 1/20 0.36
MGAM2 Q2M2H8 1/20 0.36
TRPV4 Q9HBA0 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
ATM Q13315 1/20 0.35
CTDSP1 Q9GZU7 1/20 0.35
ANO1 Q5XXA6 1/20 0.34
HTR3E A5X5Y0 1/20 0.34
HTR3B O95264 1/20 0.34
HTR3A P46098 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23522173 1.00 KMT2A (0.41) KMT2AMAPTKDM4EHPGDTSHR
SCHEMBL23522175 1.00 KMT2A (0.41) KMT2AMAPTKDM4EHPGDTSHR
SCHEMBL21723894 1.00 KMT2A (0.41) KMT2AMAPTKDM4EHPGDTSHR
SCHEMBL25403243 0.89 LMNA (0.39) KMT2AMAPTKDM4EHPGDMEN1
SCHEMBL16796949 0.85 TSHR (0.38) KMT2AMAPTHPGDTSHRMEN1
SCHEMBL16796947 0.85 TSHR (0.38) KMT2AMAPTHPGDTSHRMEN1
SCHEMBL23521961 0.84 ACHE (0.41) KMT2AMAPTTSHRMEN1ALDH1A1
SCHEMBL21723924 0.84 ACHE (0.41) KMT2AMAPTTSHRMEN1ALDH1A1
SCHEMBL21723926 0.84 ACHE (0.41) KMT2AMAPTTSHRMEN1ALDH1A1
SCHEMBL23521965 0.84 ACHE (0.41) KMT2AMAPTTSHRMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12630511-B2 Benzamide derivative, preparation method therefor, and pharmaceutical composition comprising same as active ingredient for prevention or treatment of cancer KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2026-05-19 US disclosed
US-11976059-B2 Isoindolin-1-on derivative, method for preparing same, and pharmaceutical composition comprising same as effective component for preventing or treating cancer KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2024-05-07 US disclosed
CN-114630819-B Benzamide derivative for preventing or treating cancer, method for preparing the same, and pharmaceutical composition comprising the same as active ingredient 韩国化学研究院 2024-02-13 CN disclosed
CN-112839937-B Isoindolin-1-one derivatives, preparation method and application thereof 韩国化学研究院 2023-08-22 CN disclosed
EP-3838898-B1 ISOINDOLIN-1-ONE DERIVATIVE, METHOD FOR PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME AS AN EFFECTIVE COMPONENT FOR PREVENTING OR TREATING CANCER KOREA RES INST CHEMICAL TECH (KR) 2023-06-07 EP disclosed
US-20220281817-A1 BENZAMIDE DERIVATIVE, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL COMPOSITION COMPRISING SAME AS ACTIVE INGREDIENT FOR PREVENTION OR TREATMENT OF CANCER KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2022-09-08 US disclosed
CN-114630819-A Benzamide derivatives for preventing or treating cancer, preparation method thereof, and pharmaceutical composition comprising the same as active ingredient 韩国化学研究院 2022-06-14 CN disclosed
EP-4005572-A1 BENZAMIDE DERIVATIVE, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL COMPOSITION COMPRISING SAME AS ACTIVE INGREDIENT FOR PREVENTION OR TREATMENT OF CANCER Korea Research Institute of Chemical Technology (KR) 2022-06-01 EP disclosed
US-20210332029-A1 ISOINDOLIN-1-ON DERIVATIVE, METHOD FOR PREPARING SAME, AND PHARMACEUTICAL COMPOSITION COMPRISING SAME AS EFFECTIVE COMPONENT FOR PREVENTING OR TREATING CANCER KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2021-10-28 US disclosed
EP-3838898-A1 ISOINDOLIN-1-ON DERIVATIVE, METHOD FOR PREPARING SAME, AND PHARMACEUTICAL COMPOSITION COMPRISING SAME AS EFFECTIVE COMPONENT FOR PREVENTING OR TREATING CANCER Korea Research Institute of Chemical Technology (KR) 2021-06-23 EP disclosed
CN-112839937-A Isoindolin-1-one derivative, method for preparing same, and pharmaceutical composition for preventing or treating cancer comprising same as effective component 韩国化学研究院 2021-05-25 CN disclosed
WO-2020036386-A1 ISOINDOLIN-1-ON DERIVATIVE, METHOD FOR PREPARING SAME, AND PHARMACEUTICAL COMPOSITION COMPRISING SAME AS EFFECTIVE COMPONENT FOR PREVENTING OR TREATING CANCER 한국화학연구원 2020-02-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210332029-A1 ISOINDOLIN-1-ON DERIVATIVE, METHOD FOR PREPARING SAME, AND PHARMACEUTICAL COMPOSITION COMPRISING SAME AS EFFECTIVE COMPONENT FOR PREVENTING OR TREATING CANCER EGFR, TP53, BRCA1 KMT2A 3598/4885MAPT 2651/4885KDM4E 4462/4885
US-20220281817-A1 BENZAMIDE DERIVATIVE, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL COMPOSITION COMPRISING SAME AS ACTIVE INGREDIENT FOR PREVENTION OR TREATMENT OF CANCER EGFR, WEE1, WEE2 KMT2A 1358/4885MAPT 4157/4885KDM4E 2110/4885
US-12630511-B2 Benzamide derivative, preparation method therefor, and pharmaceutical composition comprising same as active ingredient for prevention or treatment of cancer EGFR, ERBB2, KRAS KMT2A 2930/4885MAPT 4195/4885KDM4E 3236/4885
US-11976059-B2 Isoindolin-1-on derivative, method for preparing same, and pharmaceutical composition comprising same as effective component for preventing or treating cancer EGFR, TP53, BRCA1 KMT2A 3598/4885MAPT 2651/4885KDM4E 4462/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.