SCHEMBL2172564

SCHEMBL2172564

CCOc1ccc(NS(=O)(=O)c2ccccc2)cc1NC1CCN(C)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SSTR5 P35346 1/20 0.52
HRH1 P35367 1/20 0.52
HTR6 P50406 5/20 0.52
CYP3A4 P08684 2/20 0.50
MEN1 O00255 1/20 0.47
MAPT P10636 1/20 0.47
KMT2A Q03164 1/20 0.47
CYP2D6 P10635 1/20 0.46
HCRTR1 O43613 1/20 0.43
EGFR P00533 1/20 0.42
ERBB2 P04626 1/20 0.42
ERBB4 Q15303 1/20 0.42
LMNA P02545 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
SSTR4 P31391 1/20 0.41
BRD4 O60885 1/20 0.41
NSD2 O96028 1/20 0.41
HTR1A P08908 1/20 0.41
HTR7 P34969 1/20 0.41
OGG1 O15527 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2170708 0.89 HTR6 (0.63) SSTR5HRH1HTR6CYP3A4MEN1
SCHEMBL2170411 0.83 CYP3A4 (0.58) HTR6CYP3A4MEN1KMT2ACYP2D6
SCHEMBL2170725 0.83 CYP3A4 (0.50) HTR6CYP3A4MAPTLMNABRD4
SCHEMBL2183994 0.82 CYP3A4 (0.49) HTR6CYP3A4MEN1KMT2ACYP2D6
Hydrochloric Acid SCHEMBL6118475 0.81 CYP3A4 (0.48) HTR6CYP3A4MEN1KMT2ACYP2D6
SCHEMBL2172325 0.79 CYP3A4 (0.60) HRH1HTR6CYP3A4MEN1MAPT
SCHEMBL2170321 0.78 CYP3A4 (0.59) HRH1HTR6CYP3A4MEN1MAPT
SCHEMBL6118790 0.78 HTR6 (0.59) HTR6CYP3A4MEN1KMT2AL3MBTL1
SCHEMBL2170724 0.77 CYP3A4 (0.59) HRH1HTR6CYP3A4MEN1MAPT
SCHEMBL6117937 0.75 CYP3A4 (0.50) HRH1HTR6CYP3A4CYP2D6LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346847-B1 ARYL SULFONAMIDE AMINE COMPOUNDS AND THEIR USE AS 5-HT6 LIGANDS SUVEN LIFE SCIENCES LTD (IN) 2013-05-15 EP claimed
US-20120129816-A1 ARYL SULFONAMIDE AMINE COMPOUNDS AND THEIR USE AS 5-HT6 LIGANDS SUVEN LIFE SCIENCES LIMITED (IN) 2012-05-24 US claimed
EP-2346847-A1 ARYL SULFONAMIDE AMINE COMPOUNDS AND THEIR USE AS 5-HT6 LIGANDS Suven Life Sciences Limited (IN) 2011-07-27 EP claimed
WO-2010032258-A1 ARYL SULFONAMIDE AMINE COMPOUNDS AND THEIR USE AS 5-HT6 LIGANDS SUVEN LIFE SCIENCES LIMITED (IN) 2010-03-25 WO claimed
EP-2346847-B1 ARYL SULFONAMIDE AMINE COMPOUNDS AND THEIR USE AS 5-HT6 LIGANDS SUVEN LIFE SCIENCES LTD (IN) 2013-05-15 EP disclosed
US-8404720-B2 Aryl sulfonamide amine compounds and their use as 5-HT6 ligands SUVEN LIFE SCIENCES LIMITED (IN) 2013-03-26 US disclosed
US-20120129816-A1 ARYL SULFONAMIDE AMINE COMPOUNDS AND THEIR USE AS 5-HT6 LIGANDS SUVEN LIFE SCIENCES LIMITED (IN) 2012-05-24 US disclosed
EP-2346847-A1 ARYL SULFONAMIDE AMINE COMPOUNDS AND THEIR USE AS 5-HT6 LIGANDS Suven Life Sciences Limited (IN) 2011-07-27 EP disclosed
WO-2010032258-A1 ARYL SULFONAMIDE AMINE COMPOUNDS AND THEIR USE AS 5-HT6 LIGANDS SUVEN LIFE SCIENCES LIMITED (IN) 2010-03-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120129816-A1 ARYL SULFONAMIDE AMINE COMPOUNDS AND THEIR USE AS 5-HT6 LIGANDS HTR6, HTR1A, HTR5A SSTR5 28/4885HRH1 339/4885HTR6 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.