SCHEMBL21735121

SCHEMBL21735121

C=CC(=O)OCC(F)(F)OC(F)(F)OC(F)(F)OC(F)(F)CSc1ccc2cc(-c3cccnc3)oc2c1

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.32
CYP19A1 P11511 1/20 0.32
CYP2E1 P05181 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2A6 P11509 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2B6 P20813 1/20 0.32
CYP2C19 P33261 1/20 0.32
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
PGR P06401 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.30
PIM1 P11309 1/20 0.30
PIM2 Q9P1W9 1/20 0.30
MAP4K4 O95819 1/20 0.30
ABL1 P00519 1/20 0.30
NTRK1 P04629 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21735258 0.90 HDAC6 (0.36)
SCHEMBL21735118 0.89 CYP3A4 (0.33) S1PR1CYP19A1CYP2E1CYP3A4CYP2D6
SCHEMBL21734972 0.87 CYP19A1 (0.35) S1PR1CYP19A1KDM4EALDH1A1HPGD
SCHEMBL21735736 0.86 CYP2E1 (0.33) S1PR1CYP19A1CYP2E1CYP3A4CYP2D6
SCHEMBL21734967 0.86 S1PR1 (0.32) S1PR1CYP19A1CYP2E1CYP3A4CYP2D6
SCHEMBL21734932 0.85 CYP2E1 (0.34) S1PR1CYP19A1CYP2E1CYP3A4CYP2D6
SCHEMBL21735363 0.85 CYP3A4 (0.34) S1PR1CYP19A1CYP2E1CYP3A4CYP2D6
SCHEMBL22628761 0.84 KDM4E (0.31) S1PR1CYP3A4CYP2C19KDM4EALDH1A1
SCHEMBL22628758 0.82
SCHEMBL21735262 0.82 CYP3A4 (0.32) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11014901-B2 Hydrophobic compounds for optically active devices MERCK PATENT GMBH (DE) 2021-05-25 US disclosed
EP-3583091-B1 HYDROPHOBIC COMPOUNDS FOR OPTICALLY ACTIVE DEVICES MERCK PATENT GMBH (DE) 2020-11-04 EP disclosed
US-20200055833-A1 HYDROPHOBIC COMPOUNDS FOR OPTICALLY ACTIVE DEVICES MERCK PATENT GMBH (DE) 2020-02-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200055833-A1 HYDROPHOBIC COMPOUNDS FOR OPTICALLY ACTIVE DEVICES UACA, CRYZ, TRPA1 S1PR1 3951/4885CYP19A1 2317/4885CYP2E1 3677/4885
US-11014901-B2 Hydrophobic compounds for optically active devices UACA, CRYZ, TRPA1 S1PR1 3951/4885CYP19A1 2317/4885CYP2E1 3677/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.