SCHEMBL21742890

SCHEMBL21742890

Brc1ccccc1-c1cccc(-c2ccccn2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.48
ALDH1A1 P00352 1/20 0.48
CYP2A6 P11509 1/20 0.44
KDM4E B2RXH2 2/20 0.43
LMNA P02545 2/20 0.43
CCR1 P32246 2/20 0.43
CCR5 P51681 2/20 0.43
CCR8 P51685 2/20 0.43
CYP1A2 P05177 1/20 0.43
POLB P06746 1/20 0.43
METAP1 P53582 1/20 0.43
BLM P54132 1/20 0.43
HIF1A Q16665 1/20 0.43
DOHH Q9BU89 1/20 0.43
P4HTM Q9NXG6 1/20 0.43
GRM5 P41594 6/20 0.43
HTR1A P08908 1/20 0.43
HTR7 P34969 1/20 0.43
DCTPP1 Q9H773 2/20 0.43
TP53 P04637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21698323 0.91 CYP2A6 (0.40) MAPK1ALDH1A1CYP2A6KDM4ELMNA
SCHEMBL17426491 0.87 KDM4E (0.52) MAPK1ALDH1A1CYP2A6KDM4ELMNA
SCHEMBL18015186 0.85 ALDH1A1 (0.47) MAPK1ALDH1A1CYP2A6KDM4ELMNA
SCHEMBL18015184 0.85 ALDH1A1 (0.47) MAPK1ALDH1A1CYP2A6KDM4ELMNA
SCHEMBL18015355 0.84 ALDH1A1 (0.54) MAPK1ALDH1A1CYP2A6KDM4ELMNA
SCHEMBL19500912 0.83 GRM5 (0.55) MAPK1ALDH1A1CYP2A6KDM4ELMNA
SCHEMBL29679578 0.83 KDM4E (0.62) MAPK1ALDH1A1CYP2A6KDM4ELMNA
SCHEMBL502867 0.83 KDM4E (0.62) MAPK1ALDH1A1CYP2A6KDM4ELMNA
SCHEMBL28673366 0.82 MAPK1 (0.52) MAPK1ALDH1A1CYP2A6GRM5TP53
SCHEMBL21506994 0.81 KDM4E (0.59) MAPK1ALDH1A1CYP2A6KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200055822-A1 MATERIALS FOR ORGANIC ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2020-02-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200055822-A1 MATERIALS FOR ORGANIC ELECTRONIC DEVICES PNMT, DDT, TYR MAPK1 3046/4885ALDH1A1 323/4885CYP2A6 211/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.