SCHEMBL21743085

SCHEMBL21743085

CS(=O)(=O)c1ccc(-c2ccc(F)cc2F)c(C#N)c1

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EPAS1 Q99814 1/20 0.47
PTGS2 P35354 14/20 0.46
PTGS1 P23219 3/20 0.46
SCN9A Q15858 3/20 0.43
SLC22A12 Q96S37 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12327372 0.79 EPAS1 (0.55) EPAS1PTGS2PTGS1SLC22A12
SCHEMBL2888292 0.76 EPAS1 (0.51) EPAS1PTGS2PTGS1SLC22A12
SCHEMBL4064154 0.75 EPAS1 (0.46) EPAS1PTGS2PTGS1SLC22A12
SCHEMBL13448493 0.74 PTGS2 (0.72) PTGS2PTGS1
SCHEMBL21743211 0.74 RORC (0.38) PTGS2SCN9ASLC22A12
SCHEMBL4935434 0.73 LMNA (0.53) PTGS2PTGS1
SCHEMBL10051874 0.73 EPAS1 (0.55) EPAS1PTGS2PTGS1
SCHEMBL21116203 0.73 USP8 (0.42)
SCHEMBL31245792 0.73 PSEN1 (0.43) PTGS2PTGS1SCN9A
SCHEMBL21743184 0.73 PSEN1 (0.43) PTGS2PTGS1SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020035560-A1 1-METHYL-4-[(4-PHENYLPHENYL)SULFONYLMETHYL]CYCLOHEXYANOL AND 1-METHYL-4-[[4-(2-PYRIDYL)PHENYL]SULFONYLMETHYL]CYCLOHEXANOL COMPOUNDS AND THEIR THERAPEUTIC USE Modern Biosciences Limited (GB) 2020-02-20 WO disclosed