SCHEMBL21743769

SCHEMBL21743769

CN1CCc2c(cccc2N2CCN3CCCC3C2)C1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.45
HTR6 P50406 3/20 0.45
DRD3 P35462 2/20 0.45
CXCR4 P61073 2/20 0.44
CHRM5 P08912 2/20 0.44
CHRM1 P11229 2/20 0.44
CHRM3 P20309 2/20 0.44
CHRM2 P08172 1/20 0.44
CHRM4 P08173 1/20 0.44
HRH3 Q9Y5N1 3/20 0.41
MAOA P21397 2/20 0.40
MAOB P27338 2/20 0.40
SIGMAR1 Q99720 2/20 0.39
TMEM97 Q5BJF2 1/20 0.39
HTR1A P08908 1/20 0.39
ADRA2A P08913 1/20 0.39
ADRA2B P18089 1/20 0.39
ADRA2C P18825 1/20 0.39
DRD5 P21918 1/20 0.39
HRH2 P25021 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19537630 0.81 SIGMAR1 (0.56) DRD2HTR6DRD3CHRM5CHRM1
SCHEMBL21744255 0.79 MAOA (0.53) DRD2HTR6DRD3CHRM5CHRM1
SCHEMBL21744701 0.79 CXCR4 (0.48) DRD2HTR6DRD3CXCR4CHRM5
SCHEMBL21743767 0.79 CXCR4 (0.48) DRD2HTR6DRD3CXCR4CHRM5
SCHEMBL8219651 0.72 MAOA (0.47) DRD2HTR6DRD3CHRM5CHRM1
SCHEMBL21744258 0.72 HTR6 (0.52) DRD2HTR6DRD3MAOAMAOB
SCHEMBL12853760 0.71 DRD3 (0.60) DRD2HTR6DRD3MAOAMAOB
SCHEMBL24975339 0.71 CXCR4 (0.60) CXCR4CHRM5CHRM1CHRM3CHRM2
SCHEMBL23122959 0.70 MAP4K4 (0.43) HRH3TMEM97HTR2B
SCHEMBL23123116 0.67 HRH3 (0.47) HTR6HRH3ADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230112832-A1 Chemokine CXCR4 Receptor Modulators and Uses Related Thereto UNIV EMORY (US) 2023-04-13 US disclosed
US-20200054623-A1 Chemokine CXCR4 Receptor Modulators and Uses Related Thereto EMORY UNIVERSITY 2020-02-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200054623-A1 Chemokine CXCR4 Receptor Modulators and Uses Related Thereto CXCR4, CXCL12, CXCR1 DRD2 4147/4885HTR6 1689/4885DRD3 3970/4885
US-20230112832-A1 Chemokine CXCR4 Receptor Modulators and Uses Related Thereto CXCR4, CXCL12, CXCR1 DRD2 4147/4885HTR6 1689/4885DRD3 3970/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.