SCHEMBL2174470

SCHEMBL2174470

CCc1cc(NC(=O)Cc2ccc(Oc3ccnc4cc(C(=O)NC)ccc34)cc2OC)n[nH]1

nearest known ligand 0.82

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 19/20 0.82
CSF1R P07333 16/20 0.82
KDR P35968 15/20 0.82
FLT3 P36888 8/20 0.82
MET P08581 2/20 0.59
PDGFRA P16234 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2174542 0.83 PDGFRB (0.84) PDGFRBCSF1RKDRFLT3MET
SCHEMBL5598739 0.80 PDGFRB (0.74) PDGFRBCSF1RKDRFLT3MET
SCHEMBL2172536 0.78 KDR (0.81) PDGFRBCSF1RKDRFLT3MET
SCHEMBL4214384 0.76 PDGFRB (0.77) PDGFRBCSF1RKDRFLT3MET
SCHEMBL2174490 0.75 PDGFRB (0.69) PDGFRBCSF1RKDRFLT3MET
SCHEMBL2173785 0.74 PDGFRB (0.77) PDGFRBCSF1RKDRFLT3MET
SCHEMBL5598429 0.74 PDGFRB (0.65) PDGFRBCSF1RKDRFLT3MET
SCHEMBL2172612 0.74 PDGFRB (0.74) PDGFRBCSF1RKDRFLT3MET
SCHEMBL2172911 0.73 PDGFRB (1.00) PDGFRBCSF1RKDRFLT3MET
SCHEMBL2176706 0.73 PDGFRB (0.83) PDGFRBCSF1RKDRFLT3MET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7973164-B2 Quinoline derivatives ASTRAZENECA AB (SE) 2011-07-05 US claimed