SCHEMBL21747485

SCHEMBL21747485

O=C(Nc1ccccc1-c1cc2ccc(CN3CCN(C(=O)O)CC3)cc2o1)c1cccc2ccccc12

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.49
KDM4E B2RXH2 2/20 0.46
USP2 O75604 1/20 0.46
ALDH1A1 P00352 1/20 0.46
LMNA P02545 1/20 0.46
ALOX15 P16050 1/20 0.46
MAPK1 P28482 1/20 0.46
HSD17B10 Q99714 1/20 0.46
BCHE P06276 1/20 0.46
DRD4 P21917 8/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
POLB P06746 1/20 0.42
FAAH O00519 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20541721 0.90 KDM4E (0.52) KDM4EUSP2ALDH1A1LMNAALOX15
SCHEMBL20541856 0.89 BCHE (0.43) BACE1KDM4EALDH1A1BCHEDRD4
SCHEMBL20541987 0.89 S1PR1 (0.47) BACE1KDM4EALDH1A1BCHEDRD4
SCHEMBL20542016 0.89 BACE1 (0.44) BACE1KDM4EALDH1A1BCHEDRD4
SCHEMBL21747496 0.89 FAAH (0.44) BACE1LMNABCHEDRD4FAAH
SCHEMBL30468295 0.88 BACE1 (0.53) BACE1KDM4EBCHEDRD4MEN1
Hydrochloric Acid SCHEMBL20541653 0.88 BACE1 (0.46) BACE1BCHEDRD4
SCHEMBL20542002 0.88 MCHR1 (0.45) ALDH1A1HSD17B10DRD4MEN1KMT2A
SCHEMBL20541736 0.86 NPC1 (0.49) BCHEDRD4KMT2AFAAH
SCHEMBL20541911 0.85 SLC6A12 (0.47) BACE1KDM4EALDH1A1MAPK1BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3613735-A1 NOVEL SIRT 1 ACTIVATOR AND MEDICINAL USE THEREOF Pusan National University Industry - University Cooperation Foundation (KR) 2020-02-26 EP disclosed