SCHEMBL21753632

SCHEMBL21753632

Cc1cc(ONC(=O)CCC(C)c2ccccc2)n(-c2ccccc2)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
ATM Q13315 1/20 0.43
NTRK1 P04629 1/20 0.43
HTT P42858 2/20 0.42
TDP1 Q9NUW8 1/20 0.41
GAA P10253 2/20 0.40
P2RY1 P47900 1/20 0.40
LMNA P02545 2/20 0.40
STAT1 P42224 1/20 0.40
TSHR P16473 1/20 0.40
KCNJ6 P48051 1/20 0.40
KCNJ5 P48544 1/20 0.40
KCNJ3 P48549 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CYP1A2 P05177 1/20 0.39
MAPK1 P28482 1/20 0.39
CYP2C19 P33261 1/20 0.39
RCE1 Q9Y256 1/20 0.39
KMT2A Q03164 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28364642 0.85 ALDH1A1 (0.42) ALDH1A1L3MBTL1ATMNTRK1HTT
SCHEMBL21753627 0.84 ALDH1A1 (0.48) ALDH1A1L3MBTL1ATMNTRK1HTT
SCHEMBL21753616 0.81 ALDH1A1 (0.50) ALDH1A1L3MBTL1ATMNTRK1HTT
SCHEMBL21753653 0.81 P2RY1 (0.48) ALDH1A1L3MBTL1ATMNTRK1GAA
SCHEMBL21753629 0.79 P2RY1 (0.51) ALDH1A1L3MBTL1ATMNTRK1GAA
SCHEMBL21753656 0.76 ALDH1A1 (0.46) ALDH1A1L3MBTL1ATMNTRK1HTT
SCHEMBL28883960 0.76 ALDH1A1 (0.45) ALDH1A1L3MBTL1ATMNTRK1HTT
SCHEMBL21753644 0.74 P2RY1 (0.43) ALDH1A1L3MBTL1ATMNTRK1TDP1
SCHEMBL21753623 0.74 P2RY1 (0.43) ALDH1A1L3MBTL1ATMNTRK1TDP1
SCHEMBL21753619 0.74 NTRK1 (0.50) ALDH1A1L3MBTL1ATMNTRK1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020038279-A1 SUBSTITUTED PYRAZOLE COMPOUND, AND PREPARATION METHOD, PHARMACEUTICAL COMPOSITION, AND USE THEREOF 天津谷堆生物医药科技有限公司 2020-02-27 WO disclosed