SCHEMBL21753623

SCHEMBL21753623

CCCCCCC(C)C(=O)NOc1cc(C)nn1-c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
P2RY1 P47900 3/20 0.43
L3MBTL1 Q9Y468 2/20 0.41
ALDH1A1 P00352 2/20 0.41
NTRK1 P04629 2/20 0.41
LMNA P02545 1/20 0.41
STAT1 P42224 1/20 0.41
SOAT2 O75908 4/20 0.40
SOAT1 P35610 4/20 0.40
GAA P10253 3/20 0.40
KMT2A Q03164 2/20 0.40
ATM Q13315 1/20 0.40
MAPT P10636 3/20 0.39
TSHR P16473 1/20 0.38
KCNJ6 P48051 1/20 0.38
KCNJ5 P48544 1/20 0.38
KCNJ3 P48549 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21753644 1.00 P2RY1 (0.43) P2RY1L3MBTL1ALDH1A1NTRK1LMNA
SCHEMBL21753629 0.82 P2RY1 (0.51) P2RY1L3MBTL1ALDH1A1NTRK1LMNA
SCHEMBL21753653 0.79 P2RY1 (0.48) P2RY1L3MBTL1ALDH1A1NTRK1GAA
SCHEMBL21753627 0.78 ALDH1A1 (0.48) P2RY1L3MBTL1ALDH1A1NTRK1LMNA
SCHEMBL21753616 0.77 ALDH1A1 (0.50) P2RY1L3MBTL1ALDH1A1NTRK1LMNA
SCHEMBL21753632 0.74 ALDH1A1 (0.43) P2RY1L3MBTL1ALDH1A1NTRK1LMNA
SCHEMBL21774371 0.74 SOAT2 (0.43) L3MBTL1ALDH1A1NTRK1LMNASTAT1
SCHEMBL21774356 0.73 SOAT2 (0.46) L3MBTL1ALDH1A1NTRK1LMNASTAT1
SCHEMBL21753619 0.73 NTRK1 (0.50) P2RY1L3MBTL1ALDH1A1NTRK1LMNA
SCHEMBL21775898 0.72 SOAT2 (0.51) L3MBTL1ALDH1A1NTRK1LMNASTAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110857285-B Substituted pyrazole compound, preparation method, pharmaceutical composition and application thereof 江苏万高药业股份有限公司 2022-12-20 CN disclosed
CN-110857285-A Substituted pyrazole compound, preparation method, pharmaceutical composition and application thereof 天津谷堆生物医药科技有限公司 2020-03-03 CN disclosed
WO-2020038279-A1 SUBSTITUTED PYRAZOLE COMPOUND, AND PREPARATION METHOD, PHARMACEUTICAL COMPOSITION, AND USE THEREOF 天津谷堆生物医药科技有限公司 2020-02-27 WO disclosed