SCHEMBL21753899

SCHEMBL21753899

O=[N+]([O-])c1ccc(CO[SiH3])cc1

nearest known ligand 0.66

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.66
AKR1C3 P42330 1/20 0.58
LOXL2 Q9Y4K0 1/20 0.55
TSHR P16473 1/20 0.52
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA7 P43166 1/20 0.50
CA9 Q16790 1/20 0.50
RAB9A P51151 2/20 0.49
MAPT P10636 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
MAOB P27338 1/20 0.49
CYP2C19 P33261 2/20 0.48
ALDH1A1 P00352 1/20 0.48
POLB P06746 1/20 0.48
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL37463 0.83 IDO1 (0.70) IDO1AKR1C3LOXL2TSHRCA12
SCHEMBL8062311 0.83 IDO1 (0.70) IDO1AKR1C3LOXL2TSHRCA12
SCHEMBL293414 0.79 IDO1 (0.66) IDO1AKR1C3LOXL2TSHRCA12
SCHEMBL293415 0.79 IDO1 (0.66) IDO1AKR1C3LOXL2TSHRCA12
SCHEMBL7829129 0.79 IDO1 (0.66) IDO1AKR1C3LOXL2TSHRCA12
SCHEMBL23091915 0.79 IDO1 (0.66) IDO1AKR1C3LOXL2TSHRCA12
SCHEMBL4016592 0.79 IDO1 (0.66) IDO1AKR1C3LOXL2TSHRCA12
SCHEMBL12417032 0.79 IDO1 (0.66) IDO1AKR1C3LOXL2TSHRCA12
SCHEMBL7769668 0.79 IDO1 (0.66) IDO1AKR1C3LOXL2TSHRCA12
SCHEMBL439093 0.79 IDO1 (1.00) IDO1AKR1C3LOXL2TSHRCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113365985-B Compound with benzo-seven-membered ring structure, preparation method and application thereof 博诺康源(北京)药业科技有限公司 2022-08-12 CN disclosed
CN-113365985-A Compound with benzo seven-membered ring structure, preparation method and application thereof 博诺康源(北京)药业科技有限公司 2021-09-07 CN disclosed
CN-112616314-A Process for the preparation of (3R,5R) -7- [2- (4-fluorophenyl) -5-isopropyl-3-phenyl-4- [ (4-hydroxymethylphenylamino) carbonyl ] -pyrrol-1-yl ] -3, 5-dihydroxyheptanoic acid hemicalcium salt, intermediates therefor and process for the preparation of intermediates 大元制药株式会社 2021-04-06 CN disclosed
CN-112292414-A Cation-curable composition and method for producing cured product 迪睿合株式会社 2021-01-29 CN disclosed
CN-111518045-A Compound with benzo seven-membered ring structure, preparation method and application thereof 博诺康源(北京)药业科技有限公司 2020-08-11 CN disclosed
WO-2020156357-A1 COMPOUND HAVING BENZO SEVEN-MEMBERED RING STRUCTURE, PREPARATION METHOD THEREFOR, AND USE THEREOF 博诺康源(北京)药业科技有限公司 2020-08-06 WO disclosed
WO-2020040614-A1 PREPARATION METHOD FOR (3R,5R)-7-[2-(4-FLUROPHENYL)-5-ISOPROPYL-3-PHENYL-4-[(4-HYDROXYMETHYLPHENYLAMINO)CARBONYL]-PYRRROL-1-YL]-3,5-DIHYDROXY HEPTANOIC ACID HEMICALCIUM SALT, INTERMEDIATE USED THEREFOR, AND PREPARATION METHOD FOR INTERMEDIATE 대원제약주식회사 2020-02-27 WO disclosed