SCHEMBL21755834

SCHEMBL21755834

CN/C(=C\C=N)c1ncccc1COc1cnc(OC)cc1C=O

nearest known ligand 0.32

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 5/20 0.32
NPC1 O15118 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
HTT P42858 1/20 0.30
RAB9A P51151 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C8 P10632 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21755845 0.91 SGMS2 (0.32) CYP1A2CYP3A4CYP2C8CYP2C9CYP2C19
SCHEMBL21755852 0.88 EGLN1 (0.33) ERN1ALDH1A1MAPT
SCHEMBL21755847 0.87 ERN1 (0.33) ERN1NPC1ALDH1A1RAB9A
SCHEMBL21755806 0.87 SYK (0.34) ERN1NPC1ALDH1A1MAPTHTT
SCHEMBL21755841 0.84 ERN1 (0.32) ERN1NPC1ALDH1A1MAPTHTT
SCHEMBL15065402 0.83 PARP1 (0.39) ERN1NPC1ALDH1A1MAPTHTT
SCHEMBL21755836 0.82 SYK (0.38) ERN1NPC1ALDH1A1MAPTHTT
SCHEMBL15066126 0.82 KDM4E (0.42) ERN1NPC1ALDH1A1MAPTHTT
SCHEMBL30078095 0.82 KDM4E (0.42) ERN1NPC1ALDH1A1MAPTHTT
SCHEMBL21755839 0.81 ERN1 (0.32) ERN1NPC1ALDH1A1MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2797597-B1 SUBSTITUTED HETEROARYL ALDEHYDE COMPOUNDS AND METHODS FOR THEIR USE IN INCREASING TISSUE OXYGENATION GLOBAL BLOOD THERAPEUTICS INC (US) 2020-02-26 EP disclosed