SCHEMBL21755872

SCHEMBL21755872

CC(CN)Cc1ccccccccc1

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 6/20 0.60
SIGMAR1 Q99720 4/20 0.60
SLC6A2 P23975 2/20 0.60
MAOA P21397 1/20 0.60
SLC6A4 P31645 1/20 0.60
SLC6A3 Q01959 1/20 0.60
CYP2A6 P11509 1/20 0.60
ADORA2A P29274 1/20 0.60
ADORA1 P30542 1/20 0.60
CYP2D6 P10635 1/20 0.56
EPHX1 P07099 1/20 0.52
SLC18A2 Q05940 1/20 0.50
TRPA1 O75762 1/20 0.48
LOXL2 Q9Y4K0 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2736624 1.00 TAAR1 (0.60) TAAR1SIGMAR1SLC6A2MAOASLC6A4
SCHEMBL681082 1.00 TAAR1 (0.60) TAAR1SIGMAR1SLC6A2MAOASLC6A4
Hydrochloric Acid SCHEMBL28389719 0.98 TAAR1 (0.58) TAAR1SIGMAR1SLC6A2MAOASLC6A4
Hydrochloric Acid SCHEMBL20746142 0.98 TAAR1 (0.58) TAAR1SIGMAR1SLC6A2MAOASLC6A4
Ammonia Solution, Strong SCHEMBL11021206 0.98 TAAR1 (0.58) TAAR1SIGMAR1SLC6A2MAOASLC6A4
SCHEMBL4785594 0.85 SIGMAR1 (0.64) TAAR1SIGMAR1SLC6A2MAOASLC6A4
SCHEMBL24823756 0.82 AGXT (0.49) TAAR1SIGMAR1SLC6A2MAOASLC6A4
SCHEMBL11439744 0.82 LTA4H (0.48) MAOA
SCHEMBL11380543 0.82 SLC6A4 (0.69) TAAR1SIGMAR1SLC6A2MAOASLC6A4
SCHEMBL11440388 0.82 MAOB (0.60) SIGMAR1SLC6A2MAOASLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11008305-B2 DNA-PK inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2021-05-18 US disclosed
US-20200062732-A1 DNA-PK INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED 2020-02-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11008305-B2 DNA-PK inhibitors POLK, DTYMK, DCK TAAR1 4636/4885SIGMAR1 4343/4885SLC6A2 3423/4885
US-20200062732-A1 DNA-PK INHIBITORS POLK, DTYMK, DCK TAAR1 4636/4885SIGMAR1 4343/4885SLC6A2 3423/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.