SCHEMBL21759296

SCHEMBL21759296

COC1CN2C=CC=CC2=N1

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
POLB P06746 1/20 0.44
HPGD P15428 1/20 0.44
HSD17B10 Q99714 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4570765 0.76 KDM4E (0.47) KDM4EALDH1A1POLBHPGDHSD17B10
SCHEMBL13698339 0.68 KDM4E (0.44) KDM4EALDH1A1POLBHPGDHSD17B10
SCHEMBL6418003 0.66 ALDH1A1 (0.41) KDM4EALDH1A1POLBHPGDHSD17B10
SCHEMBL14470983 0.62 KDM4E (0.38) KDM4EALDH1A1POLBHPGDHSD17B10
SCHEMBL15128265 0.61
SCHEMBL13941293 0.61 KDM4E (0.37) KDM4EALDH1A1POLBHPGDHSD17B10
SCHEMBL21655004 0.61 KDM4E (0.40) KDM4EALDH1A1POLBHPGDHSD17B10
SCHEMBL15057332 0.60
SCHEMBL6422433 0.60 KDM4E (0.36) KDM4EALDH1A1POLBHPGDHSD17B10
SCHEMBL21759408 0.60 KDM4E (0.33) KDM4EALDH1A1POLBHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2585462-B1 FUSED HETEROCYCLIC COMPOUNDS AS PHOSPHODIESTERASES (PDES) INHIBITORS TAKEDA PHARMACEUTICALS CO (JP) 2020-02-26 EP disclosed