SCHEMBL21760974

SCHEMBL21760974

CS(=O)(=O)c1cc(Br)cc2c1OCC2

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.36
MAPT P10636 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
CYP2A6 P11509 1/20 0.35
PARP1 P09874 1/20 0.34
NR3C1 P04150 2/20 0.33
NR3C2 P08235 2/20 0.33
PGR P06401 1/20 0.33
RECQL P46063 1/20 0.32
POLB P06746 1/20 0.31
PTGS1 P23219 1/20 0.31
PTGS2 P35354 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.30
WDR5 P61964 1/20 0.30
EPHB4 P54760 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4647439 0.83 NPSR1 (0.38) NPSR1MAPTRXFP1PARP1NR3C1
SCHEMBL29469917 0.83 NPSR1 (0.36) NPSR1MAPTRXFP1PARP1NR3C1
SCHEMBL30016297 0.83 PARP1 (0.37) NPSR1MAPTRXFP1CYP2A6PARP1
SCHEMBL743679 0.83 NPSR1 (0.36) NPSR1MAPTRXFP1PARP1NR3C1
SCHEMBL16142977 0.80 MAPT (0.37) NPSR1MAPTRXFP1PARP1NR3C1
SCHEMBL21761112 0.78 NR3C1 (0.37) NPSR1MAPTRXFP1PARP1NR3C1
SCHEMBL12326401 0.73 LMNA (0.33) MAPTWDR5
SCHEMBL31394015 0.73 MAPT (0.36) NPSR1MAPTRXFP1CYP2A6PARP1
SCHEMBL6342164 0.73 MAPT (0.36) NPSR1MAPTRXFP1CYP2A6PARP1
SCHEMBL17007465 0.73 DHCR7 (0.47) NPSR1RECQLPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020040104-A1 BICYCLIC HETEROAROMATIC RING DERIVATIVE 杏林製薬株式会社 2020-02-27 WO disclosed