SCHEMBL21763363

SCHEMBL21763363

Cc1cc(C(=O)N2CCN(C)CC2)sc1-c1ccc2c(C)cccc2c1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 4/20 0.52
ATM Q13315 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
TSHR P16473 2/20 0.49
ERN1 O75460 3/20 0.47
HPGD P15428 2/20 0.46
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
KDM4E B2RXH2 1/20 0.46
KDR P35968 1/20 0.43
KMT2A Q03164 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
HTR2C P28335 1/20 0.42
MAPT P10636 1/20 0.42
TNKS O95271 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12674860 0.81 ERN1 (0.72) ATMNPSR1TSHRERN1
SCHEMBL21763645 0.75 L3MBTL1 (0.56) HRH4TSHRERN1HPGDKDM4E
SCHEMBL12675653 0.72 ERN1 (0.60) ATMNPSR1TSHRERN1HPGD
SCHEMBL12675423 0.70 ERN1 (0.71) ATMNPSR1ERN1
SCHEMBL18071180 0.69 HRH4 (1.00) HRH4TSHRHPGDNPC1RAB9A
SCHEMBL21763657 0.69 ERN1 (0.49) HRH4ERN1NPC1RAB9AKDM4E
SCHEMBL15846941 0.67 TSHR (0.45) HRH4ATMNPSR1TSHRHPGD
SCHEMBL12121414 0.66 HPGD (0.62) HRH4ERN1HPGDNPC1RAB9A
SCHEMBL9050585 0.66 MAPT (0.61) HRH4NPSR1TSHRNPC1RAB9A
SCHEMBL18904579 0.65 RIPK1 (0.81) HRH4HPGDNPC1RAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2496230-B1 IRE-1 ALPHA INHIBITORS FOSUN ORINOVE PHARMATECH INC (CN) 2020-02-26 EP disclosed