SCHEMBL21763645

SCHEMBL21763645

Cc1cccc2cc(-c3cc(C(=O)N4CCN(C)CC4)ccn3)ccc12

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.56
KDM4E B2RXH2 1/20 0.56
ERN1 O75460 2/20 0.55
ABL1 P00519 4/20 0.52
BCR P11274 4/20 0.52
PIK3CD O00329 3/20 0.50
PIK3CA P42336 3/20 0.50
KCNH2 Q12809 3/20 0.50
MTOR P42345 1/20 0.50
HPGD P15428 1/20 0.48
TSHR P16473 1/20 0.48
PARP1 P09874 2/20 0.48
RIPK1 Q13546 1/20 0.47
PIK3CB P42338 2/20 0.46
PIK3CG P48736 2/20 0.46
HRH4 Q9H3N8 1/20 0.46
ATR Q13535 1/20 0.46
TNKS O95271 1/20 0.46
ADORA2A P29274 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21763595 0.86 ERN1 (0.60) L3MBTL1KDM4EERN1ABL1BCR
SCHEMBL19961492 0.79 ERN1 (0.80) L3MBTL1KDM4EERN1
SCHEMBL13551840 0.79 ERN1 (0.56) L3MBTL1KDM4EERN1ABL1BCR
SCHEMBL21763363 0.75 HRH4 (0.52) KDM4EERN1HPGDTSHRHRH4
SCHEMBL30885229 0.74 L3MBTL1 (0.56) L3MBTL1KDM4EERN1PIK3CDPIK3CA
SCHEMBL27201480 0.74 L3MBTL1 (0.56) L3MBTL1KDM4EERN1PIK3CDPIK3CA
SCHEMBL10094624 0.73 ADORA2A (0.58) L3MBTL1KDM4EERN1HPGDTSHR
SCHEMBL10723960 0.72 HPGD (0.68) L3MBTL1KDM4EHPGDTSHR
SCHEMBL16199135 0.72 L3MBTL1 (1.00) L3MBTL1KDM4EERN1PIK3CDPIK3CA
SCHEMBL13618033 0.71 L3MBTL1 (0.61) L3MBTL1KDM4EERN1ABL1BCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2496230-B1 IRE-1 ALPHA INHIBITORS FOSUN ORINOVE PHARMATECH INC (CN) 2020-02-26 EP disclosed