SCHEMBL21766162

SCHEMBL21766162

COC(=O)c1ccc2c(c1)NC(=O)c1cc(C)cn1S2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
LMNA P02545 2/20 0.51
HTT P42858 2/20 0.47
ALOX15 P16050 5/20 0.44
POLB P06746 2/20 0.43
TP53 P04637 2/20 0.43
TDP1 Q9NUW8 2/20 0.43
THRB P10828 1/20 0.43
BLM P54132 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
TSHR P16473 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.39
RXFP1 Q9HBX9 1/20 0.39
ALOX5 P09917 1/20 0.38
MAPT P10636 2/20 0.38
HSD17B10 Q99714 4/20 0.38
HPGD P15428 2/20 0.38
MEN1 O00255 1/20 0.38
FGB P02675 1/20 0.38
HSP90AA1 P07900 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23159119 0.86 SMN1; SMN2 (0.47) ALDH1A1LMNAHTTALOX15POLB
SCHEMBL21766095 0.84 POLB (0.44) POLBTP53TDP1SMN1; SMN2RXFP1
SCHEMBL23159144 0.78 KMT2A (0.49) ALDH1A1LMNAPOLBTP53SMN1; SMN2
SCHEMBL22301309 0.76 ALDH1A1 (0.40) ALDH1A1LMNAHTTALOX15POLB
SCHEMBL23158968 0.76 MAPT (0.49) ALDH1A1POLBTP53SMN1; SMN2MAPT
SCHEMBL19984532 0.75 ALDH1A1 (0.58) ALDH1A1LMNAHTTALOX15POLB
SCHEMBL23158963 0.74 MITF (0.43) ALDH1A1LMNAHTTBLMSMN1; SMN2
SCHEMBL23158997 0.74 ALDH1A1 (0.50) ALDH1A1LMNAHTTBLML3MBTL1
SCHEMBL23159005 0.74 KMT2A (0.44) ALDH1A1HTTPOLBMAPTHPGD
SCHEMBL23159065 0.74 NPC1 (0.44) ALDH1A1SMN1; SMN2HSD17B10HPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020038456-A1 CRYSTAL FORM OF TRI-CYCLE COMPOUND AND APPLICATION THEREOF 福建广生堂药业股份有限公司 2020-02-27 WO disclosed