SCHEMBL21768445

SCHEMBL21768445

O=S1(=O)CCN(c2ncc(Br)c(C(F)(F)F)n2)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 1/20 0.43
NR1H3 Q13133 1/20 0.39
NR1H2 P55055 1/20 0.39
MTOR P42345 1/20 0.38
ATF1 P18846 1/20 0.37
NFKB1 P19838 1/20 0.37
ABL1 P00519 2/20 0.37
BCR P11274 2/20 0.37
ALDH1A1 P00352 3/20 0.37
MAPK1 P28482 1/20 0.37
ACHE P22303 1/20 0.36
TSHR P16473 1/20 0.36
HTT P42858 3/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
LMNA P02545 2/20 0.35
CNR2 P34972 2/20 0.34
KDM4E B2RXH2 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19145186 0.83 OPRL1 (0.46) OPRL1NR1H3NR1H2MTORATF1
SCHEMBL19105538 0.81 OPRL1 (0.44) OPRL1NR1H3NR1H2MTORATF1
SCHEMBL21768443 0.79 ALDH1A1 (0.58) MTORABL1BCRALDH1A1MAPK1
SCHEMBL20424636 0.78 POLB (0.42) OPRL1NR1H3NR1H2ABL1BCR
SCHEMBL21768436 0.77 OPRL1 (0.46) OPRL1NR1H3NR1H2ATF1NFKB1
SCHEMBL26341281 0.75 OPRL1 (0.40) OPRL1MTORATF1NFKB1ALDH1A1
SCHEMBL15415745 0.75 ADRB1 (0.39) OPRL1NR1H3NR1H2MTORATF1
SCHEMBL21768428 0.73 OPRM1 (0.48) OPRL1NR1H3NR1H2ATF1NFKB1
SCHEMBL4407481 0.73 PANK3 (0.39) OPRL1MTORALDH1A1ACHECYP2C19
SCHEMBL14983697 0.68 POLB (0.44) OPRL1ALDH1A1MAPK1ACHETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3722284-A1 3-((HETERO-)ARYL)-8-AMINO-2-OXO-1,3-DIAZA-SPIRO-[4.5]-DECANE DERIVATIVES Grünenthal GmbH (DE) 2020-10-14 EP disclosed
EP-3402781-B1 3-((HETERO-)ARYL)-8-AMINO-2-OXO-1,3-DIAZA-SPIRO-[4.5]-DECANE DERIVATIVES GRUENENTHAL GMBH (DE) 2020-03-04 EP disclosed