SCHEMBL2176850

SCHEMBL2176850

Cc1nc(Cl)c2c(n1)N(C)CC2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.40
HPGD P15428 4/20 0.40
LMNA P02545 3/20 0.40
GAA P10253 3/20 0.40
TP53 P04637 1/20 0.40
HTT P42858 1/20 0.40
RAD52 P43351 1/20 0.38
HTR1A P08908 1/20 0.37
DRD2 P14416 1/20 0.37
DRD4 P21917 1/20 0.37
KDM4E B2RXH2 5/20 0.35
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
GLA P06280 1/20 0.34
HSD17B10 Q99714 1/20 0.34
RCE1 Q9Y256 1/20 0.34
HTR3B O95264 1/20 0.32
HTR3A P46098 1/20 0.32
HRH4 Q9H3N8 1/20 0.32
ADRA2A P08913 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16924632 0.82 ALDH1A1 (0.41) ALDH1A1HPGDLMNAGAATP53
SCHEMBL24372865 0.76 HTR2A (0.49) ALDH1A1HPGDLMNAGAATP53
SCHEMBL29478833 0.76 HTR2A (0.49) ALDH1A1HPGDLMNAGAATP53
SCHEMBL19563082 0.76 ALDH1A1 (0.47) ALDH1A1HPGDLMNAGAATP53
SCHEMBL12408937 0.73 RAD52 (0.32) ALDH1A1RAD52KDM4EMEN1KMT2A
SCHEMBL21155386 0.72 RAD52 (0.42) ALDH1A1HPGDLMNAGAARAD52
SCHEMBL22365197 0.71 RAD52 (0.36) ALDH1A1HPGDLMNAGAARAD52
SCHEMBL23249518 0.71 ALDH1A1 (0.45) ALDH1A1HPGDLMNAGAATP53
SCHEMBL9379645 0.71 HTR1A (0.34) HTR1ADRD2DRD4KDM4EMEN1
SCHEMBL9912503 0.70 KMT2A (0.43) ALDH1A1HPGDLMNAGAATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2342191-B1 AROMATIC NITROGEN-CONTAINING 6-MEMBERED RING COMPOUNDS AND THEIR USE MITSUBISHI TANABE PHARMA CORP (JP) 2013-03-20 EP disclosed
EP-2342191-B1 AROMATIC NITROGEN-CONTAINING 6-MEMBERED RING COMPOUNDS AND THEIR USE MITSUBISHI TANABE PHARMA CORP (JP) 2013-03-20 EP disclosed
US-20110166135-A1 AROMATIC NITROGEN-CONTAINING 6-MEMBERED RING COMPOUNDS AND THEIR USE MITSUBISHI TANABE PHARMA CORPORATION (JP) 2011-07-07 US disclosed
US-20110166135-A1 AROMATIC NITROGEN-CONTAINING 6-MEMBERED RING COMPOUNDS AND THEIR USE MITSUBISHI TANABE PHARMA CORPORATION (JP) 2011-07-07 US disclosed
US-20110166135-A1 AROMATIC NITROGEN-CONTAINING 6-MEMBERED RING COMPOUNDS AND THEIR USE MITSUBISHI TANABE PHARMA CORPORATION (JP) 2011-07-07 US disclosed
WO-2010030027-A1 AROMATIC NITROGEN-CONTAINING 6-MEMBERED RING COMPOUNDS AND THEIR USE MITSUBISHI TANABE PHARMA CORPORATION (JP) 2010-03-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110166135-A1 AROMATIC NITROGEN-CONTAINING 6-MEMBERED RING COMPOUNDS AND THEIR USE PDE10A, PDE3A, PDE3B ALDH1A1 1520/4885HPGD 679/4885LMNA 1368/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.