SCHEMBL21769578

SCHEMBL21769578

COc1ccc(Cl)c(C(=O)NCC2(C)CC3CC(C)CC(F)(C3)C2)c1

nearest known ligand 0.72

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 19/20 0.72
P2RY12 Q9H244 1/20 0.60
TYK2 P29597 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21753443 0.84 P2RX7 (1.00) P2RX7P2RY12
SCHEMBL21753384 0.79 P2RX7 (1.00) P2RX7P2RY12
SCHEMBL23949851 0.76 P2RX7 (0.85) P2RX7P2RY12
SCHEMBL4885873 0.76 P2RX7 (1.00) P2RX7P2RY12
SCHEMBL21753383 0.76 P2RX7 (1.00) P2RX7P2RY12TYK2
SCHEMBL14160451 0.73 P2RX7 (0.64) P2RX7P2RY12TYK2
SCHEMBL23949843 0.71 P2RX7 (0.85) P2RX7P2RY12TYK2
SCHEMBL21769898 0.71 P2RX7 (0.70) P2RX7P2RY12TYK2
SCHEMBL14160475 0.70 P2RX7 (0.59) P2RX7P2RY12TYK2
SCHEMBL23949849 0.70 P2RX7 (0.58) P2RX7P2RY12TYK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020037350-A1 ADAMANTANYL-SUBSTITUTED BENZAMIDE COMPOUNDS AND THEIR USE AS P2X7 RECEPTOR ANTAGONISTS THE UNIVERSITY OF SYDNEY (AU) 2020-02-27 WO disclosed