SCHEMBL21774388

SCHEMBL21774388

N=C(OC1CC(OCc2ccccc2)[C@H](OCc2ccccc2)C(COCc2ccccc2)O1)C(Cl)(Cl)Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SSTR1 P30872 1/20 0.43
SSTR2 P30874 1/20 0.43
SSTR4 P31391 1/20 0.43
SSTR3 P32745 1/20 0.43
SSTR5 P35346 1/20 0.43
NT5E P21589 1/20 0.42
BCHE P06276 1/20 0.41
ACHE P22303 1/20 0.41
PDE4D Q08499 1/20 0.41
HTR1A P08908 1/20 0.40
GJB2 P29033 2/20 0.40
TACR2 P21452 3/20 0.36
PTPN1 P18031 5/20 0.36
PTPN2 P17706 3/20 0.36
PTPN11 Q06124 3/20 0.36
CDC25B P30305 4/20 0.35
PTPN6 P29350 2/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25101131 1.00 SSTR1 (0.43) SSTR1SSTR2SSTR4SSTR3SSTR5
SCHEMBL22073748 0.93 GJB2 (0.42) SSTR1SSTR2SSTR4SSTR3SSTR5
SCHEMBL7565301 0.83 SSTR1 (0.52) SSTR1SSTR2SSTR4SSTR3SSTR5
SCHEMBL9094454 0.82 NT5E (0.46) SSTR1SSTR2SSTR4SSTR3SSTR5
SCHEMBL9094458 0.82 NT5E (0.46) SSTR1SSTR2SSTR4SSTR3SSTR5
SCHEMBL22073087 0.81 SSTR1 (0.43) SSTR1SSTR2SSTR4SSTR3SSTR5
SCHEMBL14616676 0.81 NT5E (0.57) SSTR1SSTR2SSTR4SSTR3SSTR5
SCHEMBL13129824 0.81 NT5E (0.57) SSTR1SSTR2SSTR4SSTR3SSTR5
SCHEMBL2989107 0.81 NT5E (0.57) SSTR1SSTR2SSTR4SSTR3SSTR5
SCHEMBL19204220 0.81 NT5E (0.57) SSTR1SSTR2SSTR4SSTR3SSTR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020038279-A1 SUBSTITUTED PYRAZOLE COMPOUND, AND PREPARATION METHOD, PHARMACEUTICAL COMPOSITION, AND USE THEREOF 天津谷堆生物医药科技有限公司 2020-02-27 WO disclosed