SCHEMBL21774759

SCHEMBL21774759

O=C(O)N[C@H]1CC[C@H](n2cc(C(F)F)nn2)CC1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 3/20 0.49
PSMB8 P28062 8/20 0.37
PSMB5 P28074 8/20 0.37
PSMB9 P28065 4/20 0.37
SMYD2 Q9NRG4 2/20 0.34
IDO1 P14902 3/20 0.34
ACHE P22303 1/20 0.33
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
DPP4 P27487 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21774834 1.00 SMYD3 (0.49) SMYD3PSMB8PSMB5PSMB9SMYD2
SCHEMBL30216252 0.80 ALDH1A1 (0.54) ALDH1A1DPP4
SCHEMBL21733289 0.80 ALDH1A1 (0.54) ALDH1A1DPP4
SCHEMBL21774780 0.78 SMYD3 (0.51) SMYD3PSMB8PSMB5PSMB9SMYD2
SCHEMBL17592034 0.78 SMYD3 (0.78) SMYD3PSMB8PSMB5PSMB9SMYD2
SCHEMBL17592032 0.78 SMYD3 (0.78) SMYD3PSMB8PSMB5PSMB9SMYD2
SCHEMBL21774782 0.78 SMYD3 (0.51) SMYD3PSMB8PSMB5PSMB9SMYD2
SCHEMBL21774861 0.77 SMYD3 (0.50) SMYD3PSMB8PSMB5PSMB9SMYD2
SCHEMBL21774864 0.77 SMYD3 (0.50) SMYD3PSMB8PSMB5PSMB9SMYD2
SCHEMBL21733292 0.75 SMYD3 (0.47) SMYD3IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11572362-B2 Pyrrolo[1,2-b]pyridazine derivatives GILEAD SCIENCES, INC. (US) 2023-02-07 US disclosed
US-20200071333-A1 PYRROLO[1,2-b]PYRIDAZINE DERIVATIVES GILEAD SCIENCES, INC. 2020-03-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11572362-B2 Pyrrolo[1,2-b]pyridazine derivatives CYP11B2, CYP11B1, DHPS SMYD3 4569/4885PSMB8 3483/4885PSMB5 876/4885
US-20200071333-A1 PYRROLO[1,2-b]PYRIDAZINE DERIVATIVES CYP11B2, CYP11B1, DHPS SMYD3 4569/4885PSMB8 3483/4885PSMB5 876/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.