SCHEMBL21776629

SCHEMBL21776629

O=C(NCc1ccc(F)cc1)Nc1ccc(O)c(F)c1

nearest known ligand 0.63

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.63
POLB P06746 2/20 0.63
NPC1 O15118 2/20 0.62
MAOB P27338 1/20 0.62
ALDH1A1 P00352 1/20 0.60
PRMT3 O60678 1/20 0.60
NAMPT P43490 7/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
GAA P10253 1/20 0.56
KMT2A Q03164 2/20 0.54
ERCC1 P07992 1/20 0.53
ERCC4 Q92889 1/20 0.53
MEN1 O00255 1/20 0.51
MAPT P10636 1/20 0.51
MTOR P42345 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4357696 0.89 NAMPT (0.59) RAB9APOLBNPC1MAOBNAMPT
SCHEMBL4347646 0.87 MTOR (0.70) RAB9APOLBPRMT3NAMPTSMN1; SMN2
SCHEMBL16946645 0.78 NPC1 (0.84) RAB9APOLBNPC1MAOBALDH1A1
SCHEMBL26546719 0.78 RAB9A (0.73) RAB9APOLBNPC1MAOBALDH1A1
SCHEMBL8180564 0.77 RAB9A (0.88) RAB9APOLBNPC1MAOBALDH1A1
SCHEMBL7420189 0.77 RAB9A (1.00) RAB9APOLBNPC1MAOBALDH1A1
SCHEMBL108218 0.77 ERCC1 (0.78) RAB9APOLBNPC1SMN1; SMN2KMT2A
SCHEMBL1137106 0.77 MET (0.53) POLBALDH1A1SMN1; SMN2GAAKMT2A
SCHEMBL23747565 0.77 RAB9A (0.71) RAB9APOLBNPC1MAOBALDH1A1
Hydrochloric Acid SCHEMBL322141 0.77 MEN1 (0.49) RAB9ANPC1ALDH1A1NAMPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110862398-B Urea substituted aromatic ring-linked dioxane quinazoline or quinoline compound, composition and application thereof 北京赛特明强医药科技有限公司 2021-04-06 CN disclosed
CN-110862398-A Urea substituted aromatic ring-linked dioxane quinazoline or quinoline compound, composition and application thereof 北京赛特明强医药科技有限公司 2020-03-06 CN disclosed
WO-2020042972-A1 UREA-SUBSTITUTED AROMATIC RING-LINKED DIOXANE AND QUINAZOLINE OR QUINOLINE COMPOUND, COMPOSITION AND APPLICATION THEREOF 北京赛特明强医药科技有限公司 2020-03-05 WO disclosed
WO-2020042972-A1 UREA-SUBSTITUTED AROMATIC RING-LINKED DIOXANE AND QUINAZOLINE OR QUINOLINE COMPOUND, COMPOSITION AND APPLICATION THEREOF 北京赛特明强医药科技有限公司 2020-03-05 WO disclosed