SCHEMBL21780928

SCHEMBL21780928

CC(C)Oc1ccc(C(Br)C(=O)c2ccc(O)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.51
PARP10 Q53GL7 1/20 0.50
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
CA14 Q9ULX7 1/20 0.44
MAPT P10636 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42
ALDH1A1 P00352 2/20 0.42
POLB P06746 1/20 0.41
MEN1 O00255 2/20 0.40
MITF O75030 1/20 0.40
ACACB O00763 3/20 0.40
NPC1 O15118 1/20 0.40
HPGD P15428 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ACACA Q13085 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11566750 0.94 KMT2A (0.58) KMT2APARP10MAPTNPSR1ALDH1A1
SCHEMBL3102478 0.88 ALDH1A1 (0.53) KMT2APARP10CA1CA2MAPT
SCHEMBL5527403 0.83 KMT2A (0.46) KMT2APARP10MAPTNPSR1ALDH1A1
SCHEMBL2936991 0.81 CA12 (0.37) KMT2APARP10CA12CA1CA2
SCHEMBL5747150 0.79 KMT2A (0.63) KMT2APARP10MAPTALDH1A1POLB
SCHEMBL5943354 0.79 KMT2A (0.63) KMT2APARP10CA12CA1CA2
SCHEMBL3089210 0.77 ALDH1A1 (0.62) KMT2APARP10CA1CA2MAPT
Hydroquinone SCHEMBL8984334 0.77 KMT2A (0.85) KMT2APARP10CA12CA1CA2
SCHEMBL7855318 0.77 ALOX15 (0.48) KMT2ACA12CA1CA2CA7
SCHEMBL28485 0.76 KMT2A (0.56) KMT2APARP10CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233828-B1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF HOFFMANN LA ROCHE (CH) 2020-03-04 EP disclosed