SCHEMBL21780933

SCHEMBL21780933

COc1ccc(-c2snc(-c3ccccc3Cl)c2C(O)OC)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 3/20 0.41
HSP90AB1 P08238 3/20 0.41
LMNA P02545 2/20 0.37
NPSR1 Q6W5P4 1/20 0.37
PTGS2 P35354 1/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
PIK3CD O00329 2/20 0.37
GPBAR1 Q8TDU6 1/20 0.37
PTPN1 P18031 1/20 0.36
ALOX5 P09917 3/20 0.36
MITF O75030 1/20 0.35
MAPT P10636 1/20 0.35
PKM P14618 1/20 0.35
MAOB P27338 1/20 0.35
AGTR1 P30556 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
APP P05067 1/20 0.35
BACE1 P56817 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17845095 0.82 HSP90AA1 (0.43) HSP90AA1HSP90AB1PTGS2NPC1RAB9A
SCHEMBL17845084 0.78 GPBAR1 (0.44) HSP90AA1HSP90AB1LMNANPSR1NPC1
SCHEMBL21780774 0.77 GPBAR1 (0.46) HSP90AA1LMNANPSR1PTGS2NPC1
SCHEMBL17845090 0.77 L3MBTL1 (0.49) HSP90AA1HSP90AB1LMNANPSR1NPC1
SCHEMBL17845139 0.70 CNR1 (0.43) HSP90AA1HSP90AB1LMNANPSR1PTGS2
SCHEMBL5681041 0.69 ABL1 (0.60) NPC1RAB9AL3MBTL1PTPN1MAPT
SCHEMBL11755156 0.66 LMNA (0.48) LMNANPSR1PTGS2NPC1RAB9A
SCHEMBL17845183 0.66 APP (0.44) PTGS2NPC1RAB9AL3MBTL1PIK3CD
SCHEMBL19123777 0.64 MAPT (0.43) PTGS2L3MBTL1ALOX5MAPTGRM1
SCHEMBL7897510 0.64 ABL1 (0.46) HSP90AA1HSP90AB1LMNANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233828-B1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF HOFFMANN LA ROCHE (CH) 2020-03-04 EP disclosed