SCHEMBL21782808

SCHEMBL21782808

CCSc1c(-c2bnc(C)n2C)nc2ccccn12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.36
KDM4E B2RXH2 4/20 0.36
DPP4 P27487 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
MAPT P10636 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HSD17B10 Q99714 1/20 0.35
TDP1 Q9NUW8 1/20 0.34
GAA P10253 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
MAPK1 P28482 2/20 0.33
ADORA3 P0DMS8 1/20 0.33
ADORA1 P30542 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25759829 0.87 KDM4E (0.36) ALDH1A1KDM4EDPP4SMN1; SMN2CYP1A2
SCHEMBL20100096 0.70 DPP4 (0.35) ALDH1A1KDM4EDPP4SMN1; SMN2CYP1A2
SCHEMBL20100107 0.69 KDM4E (0.52) ALDH1A1KDM4ESMN1; SMN2NPC1RAB9A
SCHEMBL22519128 0.69 KDM4E (0.46) ALDH1A1KDM4EDPP4SMN1; SMN2NPC1
SCHEMBL21698367 0.66 PDE10A (0.32) ALDH1A1KDM4EDPP4SMN1; SMN2CYP1A2
SCHEMBL18131807 0.66 HSD17B10 (0.33) ALDH1A1KDM4EDPP4SMN1; SMN2CYP1A2
SCHEMBL18131814 0.65 PTGS1 (0.56) ALDH1A1KDM4ESMN1; SMN2CYP1A2CYP2C9
SCHEMBL20100092 0.65 ALDH1A1 (0.34) ALDH1A1KDM4EDPP4SMN1; SMN2CYP1A2
SCHEMBL24242314 0.64 KDM4E (0.41) ALDH1A1KDM4ESMN1; SMN2NPC1MAPT
SCHEMBL21698413 0.64 ALDH1A1 (0.47) ALDH1A1KDM4ESMN1; SMN2CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3617207-A1 FUSED HETEROCYCLIC COMPOUND OR SALT THEREOF, AGRICULTURAL OR HORTICULTURAL INSECTICIDE CONTAINING EITHER COMPOUND, AND METHOD FOR USING SAID INSECTICIDE Nihon Nohyaku Co., Ltd. (JP) 2020-03-04 EP disclosed