SCHEMBL21783262

SCHEMBL21783262

CCCn1cc(C(=O)O)c(=O)c2cc(F)c(N3CCN(C)CC3)c(F)c21

nearest known ligand 0.86

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 11/20 0.86
DRD3 P35462 1/20 0.60
ADRA2B P18089 1/20 0.59
MAPK1 P28482 1/20 0.59
ALDH1A1 P00352 8/20 0.59
HPGD P15428 7/20 0.59
HSD17B10 Q99714 6/20 0.59
PMP22 Q01453 1/20 0.58
ALB P02768 1/20 0.56
HRH3 Q9Y5N1 1/20 0.56
TUBB4A P04350 1/20 0.56
POLB P06746 1/20 0.56
TUBB P07437 1/20 0.56
TUBA3C P0DPH7 1/20 0.56
TUBA1B P68363 1/20 0.56
TUBA4A P68366 1/20 0.56
TUBB4B P68371 1/20 0.56
TUBB3 Q13509 1/20 0.56
TUBB2A Q13885 1/20 0.56
TUBB8 Q3ZCM7 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fleroxacin SCHEMBL29377022 0.92 KDM4E (1.00) KDM4EDRD3ADRA2BMAPK1ALDH1A1
Fleroxacin SCHEMBL48145 0.92 KDM4E (1.00) KDM4EDRD3ADRA2BMAPK1ALDH1A1
SCHEMBL312380 0.92 KDM4E (0.84) KDM4EDRD3ADRA2BMAPK1ALDH1A1
Hydrochloric Acid SCHEMBL10766749 0.92 KDM4E (0.72) KDM4EDRD3ADRA2BMAPK1ALDH1A1
Fleroxacin SCHEMBL11193870 0.91 KDM4E (0.98) KDM4EDRD3ADRA2BMAPK1ALDH1A1
SCHEMBL312186 0.91 KDM4E (0.86) KDM4EDRD3ADRA2BMAPK1ALDH1A1
Fleroxacin SCHEMBL9745354 0.91 KDM4E (0.98) KDM4EDRD3ADRA2BMAPK1ALDH1A1
Fleroxacin SCHEMBL9745337 0.91 KDM4E (0.98) KDM4EDRD3ADRA2BMAPK1ALDH1A1
Fleroxacin SCHEMBL29114441 0.90 KDM4E (0.96) KDM4EDRD3ADRA2BMAPK1ALDH1A1
Hydrochloric Acid SCHEMBL11187466 0.89 KDM4E (0.68) KDM4EDRD3ADRA2BMAPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020014269-A9 BISPHOSPHONATE QUINOLONE CONJUGATES AND USES THEREOF BIOVINC, LLC. (US) 2020-03-05 WO disclosed