SCHEMBL21790490

SCHEMBL21790490

CCCC(C)(C)Nc1ccccc1F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSIP1 O75475 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.41
TAS1R3 Q7RTX0 1/20 0.40
TAS1R1 Q7RTX1 1/20 0.40
PDK1 Q15118 1/20 0.39
PDK2 Q15119 1/20 0.39
PDK3 Q15120 1/20 0.39
PDK4 Q16654 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
RAB9A P51151 4/20 0.37
ALDH1A1 P00352 3/20 0.37
NPSR1 Q6W5P4 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALOX12 P18054 1/20 0.37
NPC1 O15118 3/20 0.37
GAA P10253 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18826818 0.85 PSIP1 (0.47) PSIP1SMN1; SMN2TAS1R3TAS1R1PDK1
SCHEMBL21799552 0.78 MAPT (0.38) SMN1; SMN2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL6882803 0.78 GAA (0.40) SMN1; SMN2ALDH1A1KDM4EALOX12GAA
SCHEMBL10294025 0.76 PDK1 (0.46) PSIP1SMN1; SMN2PDK1PDK2PDK3
SCHEMBL29791321 0.76 PDK1 (0.46) PSIP1SMN1; SMN2PDK1PDK2PDK3
SCHEMBL29569965 0.75 MAPT (0.41) CYP1A2CYP3A4CYP2C9CYP2C19RAB9A
SCHEMBL21790806 0.74 KIF11 (0.37) SMN1; SMN2RAB9AALDH1A1NPC1GAA
SCHEMBL23101845 0.73 TTR (0.38) PSIP1CYP2C19ALOX12GAAL3MBTL1
SCHEMBL1453847 0.72 GAA (0.43) CYP2C19ALDH1A1NPSR1ALOX12GAA
SCHEMBL23084860 0.69 KDM4E (0.38) SMN1; SMN2CYP3A4CYP2C9RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200071308-A1 Benzene, Pyridine, and Pyridazine Derivatives ESANEX INC (US) 2020-03-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200071308-A1 Benzene, Pyridine, and Pyridazine Derivatives CDK4, P2RX4, MKI67 PSIP1 822/4885SMN1; SMN2 3208/4885TAS1R3 2363/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.