SCHEMBL21801705

SCHEMBL21801705

COC1=CC(=O)c2nc(N3CCC(C(F)(F)F)CC3)ccc2C1=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NSD2 O96028 3/20 0.49
TDP2 O95551 2/20 0.49
TRPV3 Q8NET8 2/20 0.37
IDO1 P14902 2/20 0.35
CDC25A P30304 1/20 0.35
CDC25B P30305 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.35
MAP4K4 O95819 3/20 0.34
PDE10A Q9Y233 1/20 0.33
SPR P35270 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
PAX8 Q06710 1/20 0.32
HKDC1 Q2TB90 1/20 0.32
ATG4B Q9Y4P1 1/20 0.32
ROCK2 O75116 1/20 0.32
DRD2 P14416 1/20 0.31
DRD3 P35462 1/20 0.31
KCNH2 Q12809 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21801765 0.81 NSD2 (0.52) NSD2TDP2TRPV3IDO1CDC25A
SCHEMBL29209079 0.69 MAP4K4 (0.44) TRPV3KDM4EMAPTMAP4K4PDE10A
SCHEMBL25204837 0.64 MAP4K4 (0.47) TRPV3KDM4EMAPTMAP4K4PDE10A
SCHEMBL21801731 0.64 MAP4K4 (0.40) TRPV3KDM4EMAPTMAP4K4PDE10A
SCHEMBL21801704 0.63 TDP2 (0.61) NSD2TDP2IDO1CDC25ACDC25B
SCHEMBL1644219 0.63 HRH3 (0.52) TRPV3KDM4EMAPTMAP4K4PDE10A
SCHEMBL25191131 0.62 MAP4K4 (0.48) TRPV3KDM4EMAPTMAP4K4PDE10A
SCHEMBL29218615 0.62 MAP4K4 (0.45) TRPV3KDM4EMAPTMAP4K4PDE10A
SCHEMBL25039721 0.62 TRPV3 (0.47) TRPV3KDM4EMAPTMAP4K4PDE10A
SCHEMBL25187824 0.62 MAPT (0.47) TRPV3KDM4EMAPTMAP4K4PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020055192-A2 PREPARATION METHOD FOR QUINOLINE-5, 8-DIONE DERIVATIVE WHICH IS TGASE 2 INHIBITOR 재단법인 대구경북첨단의료산업진흥재단 2020-03-19 WO disclosed