SCHEMBL21801765

SCHEMBL21801765

COC1=CC(=O)c2nc(N3CCC(F)(F)CC3)ccc2C1=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NSD2 O96028 5/20 0.52
TDP2 O95551 2/20 0.52
SCN9A Q15858 1/20 0.40
IDO1 P14902 2/20 0.38
CDC25A P30304 1/20 0.38
CDC25B P30305 1/20 0.38
ROCK2 O75116 2/20 0.36
PTGER4 P35408 1/20 0.35
TRPV3 Q8NET8 1/20 0.34
WHR1 P49842 1/20 0.34
HKDC1 Q2TB90 2/20 0.33
PAX8 Q06710 1/20 0.33
ATG4B Q9Y4P1 1/20 0.33
CNR2 P34972 1/20 0.33
G6PD P11413 1/20 0.33
DNMT1 P26358 1/20 0.33
PTPN1 P18031 1/20 0.32
PDE7A Q13946 1/20 0.32
LRRK2 Q5S007 1/20 0.31
ACACB O00763 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21801705 0.81 NSD2 (0.49) NSD2TDP2IDO1CDC25ACDC25B
SCHEMBL21801752 0.70 S100A4 (0.48) NSD2SCN9APTGER4TRPV3ACACB
SCHEMBL23375735 0.69 SCN9A (0.40) SCN9AROCK2PTGER4TRPV3WHR1
SCHEMBL21500077 0.66 ROCK2 (0.40) SCN9AROCK2PTGER4TRPV3WHR1
SCHEMBL31346994 0.66 PTPN11 (0.42) ROCK2PTGER4TRPV3WHR1
SCHEMBL30469073 0.66 OGA (0.49) SCN9AROCK2PTGER4TRPV3WHR1
SCHEMBL25331930 0.66 OGA (0.49) SCN9AROCK2PTGER4TRPV3WHR1
SCHEMBL21801704 0.65 TDP2 (0.61) NSD2TDP2IDO1CDC25ACDC25B
SCHEMBL21801763 0.65 NSD2 (0.57) NSD2TDP2IDO1CDC25ACDC25B
SCHEMBL31105491 0.63 HRH3 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020055192-A2 PREPARATION METHOD FOR QUINOLINE-5, 8-DIONE DERIVATIVE WHICH IS TGASE 2 INHIBITOR 재단법인 대구경북첨단의료산업진흥재단 2020-03-19 WO disclosed