SCHEMBL21801709

SCHEMBL21801709

COC1=C(N=[N+]=[N-])C(=O)c2nc(-c3cnc(OC)nc3)ccc2C1=O

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NSD2 O96028 2/20 0.38
G6PD P11413 2/20 0.38
DNMT1 P26358 2/20 0.38
HKDC1 Q2TB90 1/20 0.34
PADI1 Q9ULC6 1/20 0.34
PADI3 Q9ULW8 1/20 0.34
PADI4 Q9UM07 1/20 0.34
PADI2 Q9Y2J8 1/20 0.34
ATG4B Q9Y4P1 1/20 0.34
S100A4 P26447 1/20 0.32
PIK3CA P42336 5/20 0.32
MTOR P42345 5/20 0.32
SCN9A Q15858 1/20 0.32
PLAU P00749 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21801746 0.88 NSD2 (0.36) NSD2G6PDDNMT1
SCHEMBL21801757 0.81 NSD2 (0.35) NSD2G6PDDNMT1HKDC1PADI1
SCHEMBL21801727 0.80 NSD2 (0.60) NSD2G6PDDNMT1HKDC1PADI1
SCHEMBL21801773 0.79 PARP10 (0.38) NSD2G6PDDNMT1
SCHEMBL21801758 0.79 NSD2 (0.59) NSD2G6PDDNMT1HKDC1PADI1
SCHEMBL21801749 0.77 MAPT (0.39) PLAU
SCHEMBL21801902 0.77 XDH (0.41)
SCHEMBL21801715 0.74 PIM2 (0.42)
SCHEMBL21801951 0.73 NSD2 (0.38) NSD2G6PDDNMT1PADI1PADI3
SCHEMBL21801763 0.72 NSD2 (0.57) NSD2G6PDDNMT1HKDC1ATG4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020055192-A2 PREPARATION METHOD FOR QUINOLINE-5, 8-DIONE DERIVATIVE WHICH IS TGASE 2 INHIBITOR 재단법인 대구경북첨단의료산업진흥재단 2020-03-19 WO disclosed