SCHEMBL21801902

SCHEMBL21801902

COC1=C(N=[N+]=[N-])C(=O)c2nc(-c3cccc(OC(F)(F)F)c3)ccc2C1=O

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
XDH P47989 2/20 0.41
DYRK1A Q13627 5/20 0.39
PDE10A Q9Y233 1/20 0.37
TRPV3 Q8NET8 1/20 0.36
CTSS P25774 1/20 0.36
CTSK P43235 1/20 0.36
ATR Q13535 1/20 0.36
MAOB P27338 1/20 0.35
MAOA P21397 2/20 0.35
FYN P06241 2/20 0.35
PDE4B Q07343 1/20 0.35
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
MAPT P10636 1/20 0.34
CLK2 P49760 1/20 0.34
HASPIN Q8TF76 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21801750 0.83 ABL1 (0.32) TRPV3
SCHEMBL21801799 0.82 NSD2 (0.51) XDHDYRK1APDE10ATRPV3CTSS
SCHEMBL21801756 0.82 NSD2 (0.51) XDHDYRK1APDE10ATRPV3CTSS
SCHEMBL21801773 0.81 PARP10 (0.38) ATRFYNMAPT
SCHEMBL21801749 0.80 MAPT (0.39) PDE4BMAPT
SCHEMBL21801720 0.78 TDP2 (0.48) XDHDYRK1APDE10ATRPV3CTSS
SCHEMBL21801746 0.77 NSD2 (0.36)
SCHEMBL21801715 0.77 PIM2 (0.42)
SCHEMBL21801709 0.77 NSD2 (0.38)
SCHEMBL21801788 0.76 NQO1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020055192-A2 PREPARATION METHOD FOR QUINOLINE-5, 8-DIONE DERIVATIVE WHICH IS TGASE 2 INHIBITOR 재단법인 대구경북첨단의료산업진흥재단 2020-03-19 WO disclosed