SCHEMBL21801740

SCHEMBL21801740

O=C1C=C(Br)C(=O)c2nc(-c3ccnc(Cl)c3)ccc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.40
PADI1 Q9ULC6 2/20 0.40
PADI3 Q9ULW8 2/20 0.40
PADI4 Q9UM07 2/20 0.40
PADI2 Q9Y2J8 2/20 0.40
PARP10 Q53GL7 1/20 0.38
PARP11 Q9NR21 1/20 0.38
CDC7 O00311 1/20 0.36
ROCK2 O75116 1/20 0.36
MAP4K4 O95819 1/20 0.36
CDK2 P24941 1/20 0.36
MAPKAPK2 P49137 1/20 0.36
GSK3B P49841 1/20 0.36
HIPK2 Q9H2X6 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
IRAK4 Q9NWZ3 1/20 0.36
CYP19A1 P11511 1/20 0.34
CCNC P24863 1/20 0.33
CDK8 P49336 1/20 0.33
PDE4A P27815 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21801915 0.79 PARP10 (0.42) IDO1PADI1PADI3PADI4PADI2
SCHEMBL21801784 0.76 PADI1 (0.46) PADI1PADI3PADI4PADI2PDE4A
SCHEMBL21801734 0.73 PARP10 (0.42) IDO1PADI1PADI3PADI4PADI2
SCHEMBL21801713 0.69 P4HB (0.40) PADI1PADI3PADI4PADI2PDE4A
SCHEMBL21801777 0.65 PADI1 (0.64) PADI1PADI3PADI4PADI2
SCHEMBL38657570 0.64 IDO1 (0.51) IDO1PARP10PARP11CDC7ROCK2
SCHEMBL980557 0.64 IDO1 (0.51) IDO1PARP10PARP11CDC7ROCK2
SCHEMBL21801898 0.63 PADI1 (0.50) IDO1PADI1PADI3PADI4PADI2
SCHEMBL19762806 0.63 IDO1 (0.50) IDO1GSK3BCYP19A1CCNCCDK8
SCHEMBL16232294 0.63 IDO1 (0.50) IDO1PARP10PARP11CDC7ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020055192-A2 PREPARATION METHOD FOR QUINOLINE-5, 8-DIONE DERIVATIVE WHICH IS TGASE 2 INHIBITOR 재단법인 대구경북첨단의료산업진흥재단 2020-03-19 WO disclosed