SCHEMBL21801784

SCHEMBL21801784

O=C1C=C(Br)C(=O)c2nc(-c3ccccc3)ccc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PADI1 Q9ULC6 2/20 0.46
PADI3 Q9ULW8 2/20 0.46
PADI4 Q9UM07 2/20 0.46
PADI2 Q9Y2J8 2/20 0.46
PDE4A P27815 1/20 0.43
PDE4B Q07343 1/20 0.43
PDE4C Q08493 1/20 0.43
PDE4D Q08499 1/20 0.43
BACE1 P56817 3/20 0.41
PTPRC P08575 2/20 0.40
PTPN1 P18031 2/20 0.38
PTPRF P10586 1/20 0.38
CDC25B P30305 1/20 0.38
MAPT P10636 4/20 0.37
RAB9A P51151 3/20 0.37
NPC1 O15118 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
PKM P14618 1/20 0.37
MAOB P27338 1/20 0.37
AGTR1 P30556 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21801708 0.81 PADI1 (0.68) PADI1PADI3PADI4PADI2PDE4A
SCHEMBL21801740 0.76 IDO1 (0.40) PADI1PADI3PADI4PADI2PDE4A
SCHEMBL21801713 0.76 P4HB (0.40) PADI1PADI3PADI4PADI2PDE4A
SCHEMBL31460555 0.76 RAB9A (0.48) PADI1PADI3PADI4PADI2PTPRC
SCHEMBL21801716 0.75 PADI1 (0.40) PADI1PADI3PADI4PADI2PDE4A
SCHEMBL31337073 0.74 MAOB (0.42) MAPTRAB9ANPC1SMN1; SMN2PKM
SCHEMBL21801729 0.74 AURKA (0.50) CDC25BMAPTRAB9ANPC1SMN1; SMN2
SCHEMBL28987151 0.72 CDC25B (0.47) PADI1PADI3PADI4PADI2CDC25B
SCHEMBL21801789 0.72 NSD2 (0.65) PADI1PADI3PADI4PADI2PDE4B
SCHEMBL4049450 0.71 RAB9A (0.54) PADI4PTPRCMAPTRAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020055192-A2 PREPARATION METHOD FOR QUINOLINE-5, 8-DIONE DERIVATIVE WHICH IS TGASE 2 INHIBITOR 재단법인 대구경북첨단의료산업진흥재단 2020-03-19 WO disclosed