SCHEMBL21801752

SCHEMBL21801752

CC(=O)NC1=CC(=O)c2ccc(N3CCC(F)(F)CC3)nc2C1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S100A4 P26447 1/20 0.48
NSD2 O96028 2/20 0.41
PTGER4 P35408 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
TRPV3 Q8NET8 1/20 0.39
ACACB O00763 2/20 0.36
TUBB4A P04350 1/20 0.34
TUBB P07437 1/20 0.34
TUBA3C P0DPH7 1/20 0.34
TUBA1B P68363 1/20 0.34
TUBA4A P68366 1/20 0.34
TUBB4B P68371 1/20 0.34
TUBB3 Q13509 1/20 0.34
TUBB2A Q13885 1/20 0.34
TUBB8 Q3ZCM7 1/20 0.34
TUBA3E Q6PEY2 1/20 0.34
TUBA1A Q71U36 1/20 0.34
TUBA1C Q9BQE3 1/20 0.34
TUBB6 Q9BUF5 1/20 0.34
TUBB2B Q9BVA1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6294367 0.76 S100A4 (0.62) S100A4NSD2TDP1MEN1NPC1
SCHEMBL21801779 0.72 S100A4 (0.60) S100A4NSD2TDP1MEN1NPC1
SCHEMBL21801765 0.70 NSD2 (0.52) NSD2PTGER4TRPV3ACACBSCN9A
SCHEMBL5925147 0.70 S100A4 (0.58) S100A4NSD2TDP1TUBB4ATUBB
SCHEMBL29952191 0.70 S100A4 (0.58) S100A4NSD2TDP1TUBB4ATUBB
SCHEMBL21801718 0.68 S100A4 (0.58) S100A4TDP1TRPV3MEN1NPC1
SCHEMBL21801897 0.67 S100A4 (0.56) S100A4TDP1MEN1NPC1RAB9A
SCHEMBL2599397 0.66 S100A4 (1.00) S100A4NSD2TDP1MEN1NPC1
SCHEMBL21801712 0.65 S100A4 (0.57) S100A4NSD2TDP1MEN1NPC1
SCHEMBL21801722 0.65 ABL1 (0.51) S100A4TDP1TRPV3RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020055192-A2 PREPARATION METHOD FOR QUINOLINE-5, 8-DIONE DERIVATIVE WHICH IS TGASE 2 INHIBITOR 재단법인 대구경북첨단의료산업진흥재단 2020-03-19 WO disclosed