SCHEMBL21801971

SCHEMBL21801971

OB(O)Oc1cccnc1C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SSTR4 P31391 1/20 0.38
CYP2C19 P33261 1/20 0.35
HTT P42858 1/20 0.33
HSD17B10 Q99714 1/20 0.33
RBP4 P02753 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
NOTUM Q6P988 1/20 0.33
HTR1A P08908 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
GPR119 Q8TDV5 1/20 0.32
NFE2L2 Q16236 1/20 0.32
ELANE P08246 1/20 0.32
P2RY1 P47900 2/20 0.32
GRM5 P41594 1/20 0.31
DHODH Q02127 1/20 0.31
PPIA P62937 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4372362 0.76 TSHR (0.44) SSTR4HTTHSD17B10RBP4HDAC6
SCHEMBL20578143 0.76 NAPRT (0.41)
SCHEMBL876096 0.74 SSTR4 (0.43) SSTR4HTTHSD17B10RBP4HDAC6
SCHEMBL31189701 0.73 PLAU (0.33) HTTHDAC6
SCHEMBL365391 0.72 L3MBTL1 (0.43) HTTHSD17B10HDAC6ELANE
SCHEMBL29912842 0.72 L3MBTL1 (0.43) HTTHSD17B10HDAC6ELANE
SCHEMBL16741102 0.72 KDM4E (0.47) SSTR4CYP2C19HTTHSD17B10RBP4
SCHEMBL29889397 0.72 HTT (0.36) SSTR4HTTHSD17B10HDAC6ELANE
SCHEMBL956094 0.72 HTT (0.36) SSTR4HTTHSD17B10HDAC6ELANE
SCHEMBL22581475 0.72 CHRNB2 (0.41) SSTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024217500-A1 ISOQUINOLINE COMPOUND, AND PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND USE THEREOF 上海赛默罗生物科技有限公司 2024-10-24 WO disclosed
CN-118541365-A Antagonists of muscarinic acetylcholine receptor M4 范德堡大学 2024-08-23 CN disclosed
CN-116903526-A Pyridinylpyridinone compounds 思普瑞特生物科学公司 2023-10-20 CN disclosed
CN-116891431-A Pyridinylpyridinone compounds 思普瑞特生物科学公司 2023-10-17 CN disclosed
CN-111094244-B Pyridinylpyridinone compounds 思普瑞特生物科学公司 2023-07-11 CN disclosed
CN-116041321-A Pyridinamine-pyridone compounds and pyrimidinamine-pyridone compounds 思普瑞特生物科学公司 2023-05-02 CN disclosed
CN-116041320-A Pyridinamine-pyridone compounds and pyrimidinamine-pyridone compounds 思普瑞特生物科学公司 2023-05-02 CN disclosed
CN-114144230-A Macrocyclic azolopyridine derivatives as EED and PRC2 modulators 弗尔康医疗公司 2022-03-04 CN disclosed
CN-111094244-A Pyridylpyridone compounds 思普瑞特生物科学公司 2020-05-01 CN disclosed
WO-2020055192-A2 PREPARATION METHOD FOR QUINOLINE-5, 8-DIONE DERIVATIVE WHICH IS TGASE 2 INHIBITOR 재단법인 대구경북첨단의료산업진흥재단 2020-03-19 WO disclosed