SCHEMBL21806014

SCHEMBL21806014

Nc1ncccc1-c1nnn[nH]1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 2/20 0.47
MKNK2 Q9HBH9 2/20 0.47
CDK1 P06493 1/20 0.47
CDK2 P24941 1/20 0.47
MAP4K4 O95819 1/20 0.42
NOS3 P29474 1/20 0.38
NOS1 P29475 1/20 0.38
NOS2 P35228 1/20 0.38
TGFBR1 P36897 1/20 0.36
NAPRT Q6XQN6 1/20 0.34
AKT1 P31749 3/20 0.33
AKT2 P31751 1/20 0.33
IDO1 P14902 1/20 0.33
RPS6KA5 O75582 1/20 0.31
TDP2 O95551 2/20 0.31
NSD2 O96028 2/20 0.31
PAX8 Q06710 2/20 0.31
TGM2 P21980 1/20 0.31
PADI1 Q9ULC6 1/20 0.31
PADI3 Q9ULW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8112420 0.80 TDP2 (0.39) IDO1TDP2NSD2PAX8TGM2
SCHEMBL16380549 0.79 MKNK1 (0.38) MKNK1MKNK2GAA
SCHEMBL28388519 0.79 PDE5A (0.34) IDO1TDP2NSD2PAX8ABL1
SCHEMBL7212308 0.78 PRMT5 (0.35) AKT1
SCHEMBL12615990 0.76 ALDH1A1 (0.38) IDO1MEN1KMT2AGAA
SCHEMBL2627823 0.76 TNKS2 (0.34)
SCHEMBL17478606 0.76 MKNK1 (0.38) MKNK1MKNK2CDK2THRBBLM
SCHEMBL18226941 0.76 CA1 (0.34) TDP2NSD2PAX8ABL1PLCG1
SCHEMBL30940314 0.76 ALDH1A1 (0.52) IDO1TDP1GAA
SCHEMBL3277728 0.76 ALDH1A1 (0.52) IDO1TDP1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3852736-A1 FARNESOID X RECEPTOR AGONISTS AND USES THEREOF Metacrine, Inc. (US) 2021-07-28 EP disclosed
WO-2020061118-A1 FARNESOID X RECEPTOR AGONISTS AND USES THEREOF METACRINE, INC. (US) 2020-03-26 WO disclosed
WO-2020061117-A1 FARNESOID X RECEPTOR AGONISTS AND USES THEREOF METACRINE, INC. (US) 2020-03-26 WO disclosed