SCHEMBL7212308

SCHEMBL7212308

NCc1ncccc1-c1nnn[nH]1

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PRMT5 O14744 3/20 0.35
WDR77 Q9BQA1 3/20 0.35
DPP4 P27487 1/20 0.33
AKT1 P31749 1/20 0.32
ALDH1A1 P00352 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21806014 0.78 MKNK1 (0.47) AKT1
SCHEMBL6919819 0.76 DPP4 (0.47) DPP4ALDH1A1L3MBTL1
SCHEMBL8112420 0.76 TDP2 (0.39) ALDH1A1
Hydrochloric Acid SCHEMBL5855503 0.75 DPP4 (0.46) DPP4
SCHEMBL28388519 0.75 PDE5A (0.34)
SCHEMBL16380549 0.75 MKNK1 (0.38) PRMT5WDR77ALDH1A1
SCHEMBL12615990 0.72 ALDH1A1 (0.38) ALDH1A1L3MBTL1
SCHEMBL2627823 0.72 TNKS2 (0.34)
SCHEMBL18226941 0.72 CA1 (0.34)
SCHEMBL17478606 0.72 MKNK1 (0.38) ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1359913-A1 THROMBIN INHIBITORS Merck & Co., Inc. (US) 2003-11-12 EP disclosed
WO-2002064211-A1 THROMBIN INHIBITORS MERCK & CO., INC. (US) 2002-08-22 WO disclosed
WO-2002064140-A1 THROMBIN INHIBITORS MERCK & CO., INC. (US) 2002-08-22 WO disclosed
WO-2002064559-A2 THROMBIN INHIBITORS MERCK & CO., INC. (US) 2002-08-22 WO disclosed