SCHEMBL21807796

SCHEMBL21807796

c1c[nH]c([C]2CCCC2)c1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.35
KDR P35968 1/20 0.35
HDAC6 Q9UBN7 2/20 0.33
HDAC1 Q13547 1/20 0.33
TSHR P16473 1/20 0.32
PARP1 P09874 1/20 0.31
KDM4C Q9H3R0 1/20 0.31
DAO P14920 1/20 0.30
HDAC8 Q9BY41 1/20 0.30
AURKB Q96GD4 1/20 0.30
INCENP Q9NQS7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6650225 0.98 AURKA (0.34) AURKAKDRHDAC6HDAC1TSHR
SCHEMBL22807093 0.95
SCHEMBL3631373 0.90
SCHEMBL630634 0.74 HDAC6 (0.41) AURKAKDRHDAC6HDAC1TSHR
Hydrochloric Acid SCHEMBL7988951 0.72 HDAC6 (0.40) AURKAKDRHDAC6HDAC1PARP1
SCHEMBL9825294 0.72 JAK2 (0.41) AURKAKDRHDAC1
SCHEMBL2088246 0.69 ACMSD (0.38) AURKAKDRHDAC6HDAC1
SCHEMBL31187621 0.67 CHRNB4 (0.42) TSHR
SCHEMBL9419852 0.67 HDAC6 (0.57) AURKAKDRHDAC6HDAC1KDM4C
SCHEMBL380666 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3852746-A1 CYCLOPENTYL ACIDS AS LPA ANTAGONISTS Bristol-Myers Squibb Company (US) 2021-07-28 EP disclosed
WO-2020060915-A1 CYCLOPENTYL ACIDS AS LPA ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2020-03-26 WO disclosed