Methoxyphenamine

Methoxyphenamine

SCHEMBL218289

CNC(C)Cc1ccccc1OC

nearest known ligand 0.63

Full drug profile on Sugi Atlas →

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.50
SLC18A2 Q05940 1/20 0.50
SIGMAR1 Q99720 1/20 0.50
ALDH1A1 P00352 1/20 0.49
GAA P10253 1/20 0.49
MAPT P10636 1/20 0.49
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
SLC6A2 P23975 1/20 0.48
SLC6A4 P31645 1/20 0.48
SLC6A3 Q01959 1/20 0.48
KCNH2 Q12809 1/20 0.48
ATM Q13315 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
IDO1 P14902 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Methoxyphenamine SCHEMBL29390678 1.00 TAAR1 (0.50) TAAR1SLC18A2SIGMAR1ALDH1A1GAA
Methoxyphenamine SCHEMBL14655868 1.00 TAAR1 (0.50) TAAR1SLC18A2SIGMAR1ALDH1A1GAA
Methoxyphenamine SCHEMBL2751759 1.00 TAAR1 (0.50) TAAR1SLC18A2SIGMAR1ALDH1A1GAA
Methoxyphenamine SCHEMBL29379229 0.98 ALDH1A1 (0.51) TAAR1SLC18A2SIGMAR1ALDH1A1GAA
Methoxyphenamine SCHEMBL208636 0.98 ALDH1A1 (0.51) TAAR1SLC18A2SIGMAR1ALDH1A1GAA
SCHEMBL20545745 0.84 ALDH1A1 (0.53) ALDH1A1GAACYP3A4CYP2D6L3MBTL1
SCHEMBL4031642 0.83 IDO1 (0.51) ALDH1A1GAAMAPTCYP3A4CYP2D6
SCHEMBL11743782 0.82 SIGMAR1 (0.53) TAAR1SIGMAR1ALDH1A1GAAMAPT
Methoxyphenamine SCHEMBL6625653 0.82 ALDH1A1 (0.53) ALDH1A1GAAMAPTCYP3A4CYP2D6
SCHEMBL878976 0.80 IDO1 (0.53) TAAR1SIGMAR1ALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2021 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4722714-A1 SIMULTANEOUS ANALYSIS OF FOOD-BORNE DOPING SUBSTANCES USING LIQUID CHROMATOGRAPHY-MASS SPECTROMETRY (VFD: VACCINE FOR FOODBORNE DOPING) Korea Institute of Science and Technology (KR) 2026-04-08 EP claimed
US-20260027139-A1 TREATMENT OF SLEEP APNEA WITH A COMBINATION OF A CARBONIC ANHYDRASE INHIBITOR AND AN ALDOSTERONE ANTAGONIST VIVUS, INC. 2026-01-29 US claimed
US-20250213647-A1 CHEMOKINE RECEPTORS AND ALPHA1 ADRENERGIC RECEPTORS/VASOPRESSIN RECEPTORS 1A HETEROMERS AS DRUG TARGETS FOR DISEASE UNIVERSITY OF SOUTH FLORIDA 2025-07-03 US claimed
US-20250017878-A1 USE OF NADOLOL TO TREAT CHRONIC OBSTRUCTIVE PULMONARY DISEASE BY BLOCKAGE OF THE ARRESTIN-2 PATHWAY CHRONIC AIRWAY THERAPEUTICS LTD (AU) 2025-01-16 US claimed
CN-119233997-A Tetrahedral antibodies 生物分子控股有限责任公司 2024-12-31 CN claimed
US-20240398729-A1 Methods and Compositions for the Treatment of Cytoplasmic Glycogen Storage Disorders DUKE UNIVERSITY (US) 2024-12-05 US claimed
EP-4463485-A2 TETRAHEDRAL ANTIBODIES Biomolecular Holdings LLC (US) 2024-11-20 EP claimed
US-12099052-B2 Method for detecting human ingested substance and ingestion times XIAMEN LISI TECH SERVICE CO., LTD. (CN) 2024-09-24 US claimed
WO-2024189434-A1 USE OF NADOLOL TO TREAT PULMONARY SYMPTOMS ASSOCIATED WITH INFECTIONS WITH SARS-CoV-2 CHRONIC AIRWAY THERAPEUTICS LIMITED (AU) 2024-09-19 WO claimed
US-20240139224-A1 TREATMENT OF SLEEP APNEA WITH A COMBINATION OF A CARBONIC ANHYDRASE INHIBITOR AND AN ALDOSTERONE ANTAGONIST AMERICAN ENTERTAINMENT PROPERTIES CORP., AS LENDER 2024-05-02 US claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
EP-0580860-B1 METHOD OF MANUFACTURING SOLID DISPERSION NIPPON SHINYAKU CO LTD (JP) 1997-10-22 EP claimed
WO-1997004764-A1 TOPICAL PHENYLEPHRINE PREPARATION ARMSTRONG KENNETH T (CA) 1997-02-13 WO claimed
EP-0724450-A1 COMPOSITION FOR WEIGHT REDUCTION CONTAINING EPHEDRINE AND A MINERAL SALT OR CHELATE Keown, Wendy J. (US) 1996-08-07 EP claimed
US-5543405-A MIXTURE OF EPHEDRINE AND CHROMIUM PICOLINATE KEOWN WENDY J (US) 1996-08-06 US claimed
WO-1995011034-A1 COMPOSITION FOR WEIGHT REDUCTION CONTAINING EPHEDRINE AND A MINERAL SALT OR CHELATE KEOWN WENDY J (US) 1995-04-27 WO claimed
EP-0311383-B1 MONOCLONAL ANTIBODY TO METHAMPHETAMINE, PREPARATION OF THE SAME, ASSAY METHOD AND ASSAY KIT OF METHAMPHETAMINE UBE INDUSTRIES, LTD. (JP) 1993-10-06 EP claimed
US-4885312-A Method for enhancing the effect of indirect-acting sympathomimetic amines MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 1989-12-05 US claimed
EP-0152379-A2 Process for preparing pharmaceutical compositions containing unilamellar liposomes CIBA-GEIGY AG (CH) 1985-08-21 EP claimed
US-RE29875-E THEOPHYLLINE SOLUBILIZED BY GLYCERYL GUAIACOLATE, POTASSIUM GUAIACOL SULFONATE OR GUAIACOL MEAD JOHNSON & COMPANY (US) 1979-01-02 US claimed