SCHEMBL21845822

SCHEMBL21845822

Cc1ccc(N2CCCN(c3ccc(C)cc3Cl)CC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
LMNA P02545 3/20 0.45
MAPK1 P28482 2/20 0.45
GFER P55789 2/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
ALDH1A1 P00352 4/20 0.45
POLB P06746 2/20 0.45
ADRB1 P08588 1/20 0.44
MAPT P10636 6/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
GAA P10253 2/20 0.43
DHFR P00374 1/20 0.43
ALDH1A3 P47895 1/20 0.42
KDM4E B2RXH2 2/20 0.41
RAD52 P43351 1/20 0.41
S100B P04271 1/20 0.41
TP53 P04637 1/20 0.41
CHRM2 P08172 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12908043 0.86 ALDH1A1 (0.58) MEN1KMT2ALMNAMAPK1ALDH1A1
SCHEMBL13419187 0.84 ALDH1A1 (0.61) MEN1KMT2ALMNAMAPK1ALDH1A1
SCHEMBL13907868 0.83 MAPT (0.57) KMT2ANPC1RAB9AALDH1A1POLB
SCHEMBL18118476 0.80 ADRB1 (0.64) MEN1KMT2ALMNANPC1RAB9A
SCHEMBL12082638 0.79 MAPT (0.64) LMNAMAPK1NPC1RAB9AALDH1A1
SCHEMBL12864867 0.77 MAPT (0.64) MEN1KMT2ALMNAMAPK1NPC1
SCHEMBL12772282 0.77 CHRM1 (0.51) MEN1KMT2ALMNANPC1RAB9A
SCHEMBL13419460 0.75 HTR3A (0.56) ADRB1
SCHEMBL327765 0.75 ADRB1 (0.64) MEN1KMT2ALMNANPC1RAB9A
SCHEMBL10063748 0.75 ADRB1 (0.70) MEN1KMT2ALMNAMAPK1GFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3626242-A1 ITRACONAZOLE ANALOGS AS INHIBITORS OF FIBROSIS The Scripps Research Institute (US) 2020-03-25 EP disclosed