SCHEMBL2184835

SCHEMBL2184835

CC(C)(C)OC(=O)[C@@]1(COc2cncc(-c3cc(F)cc(CCCO)c3)c2)CCN1

nearest known ligand 0.33

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.33
CHRNA4 P43681 2/20 0.33
NR1H2 P55055 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2185728 0.87 BACE1 (0.34) CHRNB2CHRNA4NR1H2
SCHEMBL3358712 0.76 AKT1 (0.38) NR1H2
SCHEMBL2184837 0.76 CHRNB2 (0.41) CHRNB2CHRNA4
SCHEMBL2300520 0.75 DGAT1 (0.37) CHRNB2CHRNA4
SCHEMBL2185911 0.75 DGAT1 (0.37) CHRNB2CHRNA4
SCHEMBL2185542 0.73 AKT1 (0.36) CHRNB2CHRNA4
SCHEMBL2184886 0.73 SLC5A1 (0.31)
SCHEMBL2307750 0.73 AKT1 (0.38) CHRNB2CHRNA4
SCHEMBL2185799 0.71 CHRNB2 (0.61) CHRNB2CHRNA4
Hydrochloric Acid SCHEMBL3356520 0.71 CHRNB2 (0.62) CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2342192-A2 NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS AND THE USES THEREOF Psychogenics Inc. (US) 2011-07-13 EP disclosed
WO-2010045212-A2 NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS AND THE USES THEREOF PSYCHOGENICS, INCSTATUTS (US) 2010-04-22 WO disclosed