SCHEMBL2185644

SCHEMBL2185644

Cc1nc(C(N)=O)c(-c2ccccc2C(F)(F)F)s1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 5/20 0.47
PARP1 P09874 1/20 0.45
CDC7 O00311 1/20 0.43
CCNE1 P24864 1/20 0.43
CDK2 P24941 1/20 0.43
DBF4 Q9UBU7 1/20 0.43
ALDH1A1 P00352 2/20 0.43
HPGD P15428 1/20 0.43
HCRTR1 O43613 5/20 0.42
HCRTR2 O43614 5/20 0.42
HSD11B1 P28845 2/20 0.42
NPC1 O15118 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
NTRK1 P04629 1/20 0.41
SCN10A Q9Y5Y9 1/20 0.40
KMO O15229 1/20 0.39
TRPA1 O75762 1/20 0.39
TRPM8 Q7Z2W7 1/20 0.39
TRPV1 Q8NER1 1/20 0.39
MPL P40238 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL269412 0.88 ALDH1A1 (0.50) SCN9AALDH1A1HPGDHCRTR1HCRTR2
SCHEMBL269335 0.84 ALDH1A1 (0.47) SCN9AALDH1A1HPGDHCRTR1HCRTR2
SCHEMBL327579 0.78 HSD11B1 (0.47) ALDH1A1HSD11B1NPC1TRPA1TRPM8
SCHEMBL1572631 0.77 HCRTR1 (0.43) HCRTR1HCRTR2
SCHEMBL1572629 0.77 HCRTR1 (0.43) HCRTR1HCRTR2
SCHEMBL2189924 0.77 IKBKB (0.53) PARP1CDC7ALDH1A1HPGDHCRTR1
SCHEMBL2931884 0.76 HCRTR1 (0.47) HCRTR1HCRTR2
SCHEMBL3827319 0.75 HCRTR1 (0.41) HCRTR1HCRTR2
SCHEMBL19233127 0.74 GPR52 (0.42) ALDH1A1HPGDHCRTR1HCRTR2HSD11B1
SCHEMBL1572633 0.74 HCRTR1 (0.45) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7973061-B2 Anaplastic lymphoma kinase modulators and methods of use EXELIXIS, INC. (US) 2011-07-05 US disclosed
US-20090186905-A1 ANAPLASTIC LYMPHOMA KINASE MODULATORS AND METHODS OF USE EXELIXIS, INC. (US) 2009-07-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090186905-A1 ANAPLASTIC LYMPHOMA KINASE MODULATORS AND METHODS OF USE ALK, BCL3, MCL1 SCN9A 3628/4885PARP1 768/4885CDC7 565/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.