SCHEMBL2185877

SCHEMBL2185877

NCc1cccc(-c2cncc(OC[C@]3(C(=O)OCc4ccccc4)CCN3)c2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFD P00746 2/20 0.44
PLAU P00749 4/20 0.38
PLG P00747 2/20 0.38
F11 P03951 1/20 0.38
KLKB1 P03952 1/20 0.38
F7 P08709 1/20 0.38
TPSB2 P20231 1/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNA4 P43681 1/20 0.38
MEN1 O00255 1/20 0.38
HTT P42858 1/20 0.38
GFER P55789 1/20 0.38
KMT2A Q03164 1/20 0.38
HSD17B10 Q99714 1/20 0.38
AKT1 P31749 3/20 0.38
ABL1 P00519 1/20 0.38
CYP4F2 P78329 1/20 0.35
CYP4A11 Q02928 1/20 0.35
NR4A2 P43354 1/20 0.35
MRGPRX4 Q96LA9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2186288 0.90 CYP4F2 (0.40) CFDCHRNB2CHRNA4MEN1HTT
SCHEMBL2185662 0.79 MEN1 (0.40) MEN1HTTGFERKMT2AHSD17B10
SCHEMBL2184830 0.77 CHRNB2 (0.40) CHRNB2CHRNA4MEN1HTTGFER
SCHEMBL2307750 0.75 AKT1 (0.38) CHRNB2CHRNA4AKT1ABL1
SCHEMBL2185728 0.74 BACE1 (0.34) CHRNB2CHRNA4AKT1CYP4F2CYP4A11
SCHEMBL2185883 0.74 CHRNB2 (0.47) CFDCHRNB2CHRNA4ABL1
SCHEMBL7409828 0.74 P4HTM (0.41)
SCHEMBL2185542 0.72 AKT1 (0.36) CHRNB2CHRNA4AKT1
SCHEMBL7412039 0.72 P4HTM (0.39)
SCHEMBL3358712 0.70 AKT1 (0.38) AKT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2342192-A2 NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS AND THE USES THEREOF Psychogenics Inc. (US) 2011-07-13 EP disclosed
WO-2010045212-A2 NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS AND THE USES THEREOF PSYCHOGENICS, INCSTATUTS (US) 2010-04-22 WO disclosed