SCHEMBL2184830

SCHEMBL2184830

O=C(OCc1ccccc1)[C@@]1(COc2cncc(N3CC4CC4C3)c2)CCN1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.40
CHRNA4 P43681 3/20 0.40
CHRNB4 P30926 4/20 0.39
CHRNA3 P32297 4/20 0.39
MEN1 O00255 1/20 0.39
HTT P42858 1/20 0.39
GFER P55789 1/20 0.39
KMT2A Q03164 1/20 0.39
HSD17B10 Q99714 1/20 0.39
GRIN2B Q13224 1/20 0.36
DDB1 Q16531 1/20 0.35
CRBN Q96SW2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2185662 0.80 MEN1 (0.40) MEN1HTTGFERKMT2AHSD17B10
SCHEMBL2185877 0.77 CFD (0.44) CHRNB2CHRNA4MEN1HTTGFER
SCHEMBL2186288 0.76 CYP4F2 (0.40) CHRNB2CHRNA4CHRNB4CHRNA3MEN1
SCHEMBL2184832 0.76 SIGMAR1 (0.44) CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL7409828 0.74 P4HTM (0.41) DDB1CRBN
SCHEMBL7412039 0.73 P4HTM (0.39) DDB1CRBN
SCHEMBL23199749 0.71 CHRNB2 (0.67) CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL1134480 0.71 CHRNB2 (0.67) CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL652088 0.69 GPR119 (0.48) CHRNB2CHRNA4
SCHEMBL652089 0.69 GPR119 (0.48) CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2342192-A2 NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS AND THE USES THEREOF Psychogenics Inc. (US) 2011-07-13 EP disclosed
WO-2010045212-A2 NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS AND THE USES THEREOF PSYCHOGENICS, INCSTATUTS (US) 2010-04-22 WO disclosed