SCHEMBL2186288

SCHEMBL2186288

O=C(OCc1ccccc1)[C@@]1(COc2cncc(-c3cccc(CCO)c3)c2)CCN1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 2/20 0.40
CYP4A11 Q02928 2/20 0.40
CHRNB2 P17787 2/20 0.37
CHRNA4 P43681 2/20 0.37
MEN1 O00255 1/20 0.37
HTT P42858 1/20 0.37
GFER P55789 1/20 0.37
KMT2A Q03164 1/20 0.37
HSD17B10 Q99714 1/20 0.37
CDK8 P49336 1/20 0.37
AKT1 P31749 3/20 0.36
SLC5A1 P13866 2/20 0.35
ACMSD Q8TDX5 1/20 0.35
NR4A2 P43354 1/20 0.34
MRGPRX4 Q96LA9 1/20 0.34
DDB1 Q16531 1/20 0.34
CRBN Q96SW2 1/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNA7 P36544 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2185877 0.90 CFD (0.44) CYP4F2CYP4A11CHRNB2CHRNA4MEN1
SCHEMBL2185728 0.81 BACE1 (0.34) CYP4F2CYP4A11CHRNB2CHRNA4CDK8
SCHEMBL2185662 0.79 MEN1 (0.40) MEN1HTTGFERKMT2AHSD17B10
SCHEMBL2184830 0.76 CHRNB2 (0.40) CHRNB2CHRNA4MEN1HTTGFER
SCHEMBL2307750 0.75 AKT1 (0.38) CHRNB2CHRNA4CDK8AKT1
SCHEMBL2186290 0.74 CHRNB2 (0.46) CYP4F2CYP4A11CHRNB2CHRNA4CHRNB4
SCHEMBL2185542 0.74 AKT1 (0.36) CHRNB2CHRNA4AKT1SLC5A1CHRNB4
SCHEMBL3358712 0.73 AKT1 (0.38) AKT1SLC5A1
SCHEMBL7409828 0.73 P4HTM (0.41) DDB1CRBN
SCHEMBL7412039 0.71 P4HTM (0.39) DDB1CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2342192-A2 NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS AND THE USES THEREOF Psychogenics Inc. (US) 2011-07-13 EP disclosed
WO-2010045212-A2 NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS AND THE USES THEREOF PSYCHOGENICS, INCSTATUTS (US) 2010-04-22 WO disclosed