SCHEMBL21865286

SCHEMBL21865286

Oc1ccc2cc(N3CCOCC3)ccc2c1F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 1/20 0.52
HSD17B2 P37059 1/20 0.52
PRKDC P78527 5/20 0.48
MAPT P10636 3/20 0.48
PIK3CD O00329 3/20 0.48
PIK3CA P42336 3/20 0.48
PIK3CB P42338 3/20 0.48
KDM4E B2RXH2 2/20 0.48
HTT P42858 2/20 0.48
PIK3CG P48736 2/20 0.48
NSD2 O96028 1/20 0.48
LMNA P02545 1/20 0.48
TSHR P16473 1/20 0.48
CASP1 P29466 1/20 0.48
CASP7 P55210 1/20 0.48
CASP6 P55212 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
PKM P14618 1/20 0.46
ESR1 P03372 1/20 0.45
ESR2 Q92731 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13551836 0.80 HSD17B1 (0.50) HSD17B1HSD17B2PRKDCMAPTPIK3CD
SCHEMBL13551903 0.79 ERN1 (0.63) HSD17B1HSD17B2PRKDCMAPTPIK3CD
SCHEMBL11791151 0.76 PRKDC (0.65) HSD17B1HSD17B2PRKDCMAPTPIK3CD
SCHEMBL4649483 0.74 MAPT (0.59) HSD17B1HSD17B2PRKDCMAPTPIK3CD
SCHEMBL13551847 0.73 MAPT (0.49) HSD17B1HSD17B2PRKDCMAPTPIK3CD
SCHEMBL21865069 0.73 TSHR (0.46) HSD17B1HSD17B2PRKDCMAPTPIK3CA
SCHEMBL19381145 0.73 LGMN (0.64) PRKDCMAPTPIK3CDPIK3CAPIK3CB
SCHEMBL13551895 0.71 PRKDC (0.59) HSD17B1HSD17B2PRKDCMAPTPIK3CD
SCHEMBL23693734 0.71 PRKDC (0.55) PRKDCMAPTPIK3CDPIK3CAPIK3CB
SCHEMBL3047397 0.71 LGMN (0.62) HSD17B1HSD17B2PRKDCMAPTPIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020063854-A1 QUINOLINE-BASED DERIVATIVES AS VAP-1 INHIBITORS 南京明德新药研发有限公司 2020-04-02 WO disclosed